CAS 1261392-55-5

Asenapine-13C-D3 hydrochloride

Description:

Asenapine-13C-D3 hydrochloride is a labeled derivative of asenapine, an atypical antipsychotic used primarily in the treatment of schizophrenia and bipolar disorder. The "13C-D3" designation indicates that this compound contains isotopes of carbon and deuterium, which are often used in research to trace metabolic pathways and study pharmacokinetics. Asenapine acts primarily as an antagonist at various neurotransmitter receptors, including serotonin and dopamine receptors, contributing to its therapeutic effects. The hydrochloride form enhances the solubility and stability of the compound in aqueous solutions, making it suitable for pharmaceutical formulations. Characteristically, asenapine exhibits a complex structure with multiple functional groups, which contribute to its pharmacological activity. The compound is typically administered sublingually, allowing for rapid absorption and onset of action. Safety and efficacy profiles are well-documented, but like all medications, it may have side effects and contraindications that should be considered in clinical use.

Formula: C₁₇H₁₃ClD₃NO·ClH

Synonyms:

• (3aR,12bR)-5-Chloro-2-(methyl-13C-d3)-2,3,3a,12b-tetrahydro-1H-dibenzo[2,3:6,7]oxepino[4,5-c]pyrrole hydrochloride
• Asenapine-13C-D3 hydrochloride
• [13C,2H3]-Asenapine hydrochloride

Asenapine-13C-d3 HCl

CAS: 1261392-55-5

Formula: C₁₆₁₃CH₁₃D₃ClNO·HCl

Color and Shape: White To Off-White Solid

Molecular weight: 289.78 36.46

Ref: 4Z-A-502