CAS 129029-23-8

Ocaperidone

Description:

Ocaperidone is an atypical antipsychotic medication primarily used in the treatment of schizophrenia and other psychiatric disorders. It belongs to the class of compounds known as benzisoxazoles, which are characterized by their unique bicyclic structure. The chemical formula of ocaperidone reflects its complex molecular architecture, contributing to its pharmacological properties. This substance acts as a dopamine D2 receptor antagonist, which helps to modulate neurotransmitter activity in the brain, thereby alleviating symptoms associated with psychotic disorders. Additionally, ocaperidone exhibits affinity for serotonin receptors, which may enhance its therapeutic effects and reduce side effects commonly associated with traditional antipsychotics. Its pharmacokinetic profile includes oral bioavailability, and it is metabolized in the liver, with various metabolites contributing to its overall efficacy and safety. As with many antipsychotic medications, ocaperidone may have side effects, including metabolic changes and extrapyramidal symptoms, necessitating careful monitoring during treatment. Overall, ocaperidone represents a significant advancement in the pharmacotherapy of schizophrenia, offering a balance between efficacy and tolerability.

Formula: C₂₄H₂₅FN₄O₂

InChI: InChI=1/C24H25FN4O2/c1-15-4-3-10-29-23(15)26-16(2)19(24(29)30)9-13-28-11-7-17(8-12-28)22-20-6-5-18(25)14-21(20)31-27-22/h3-6,10,14,17H,7-9,11-13H2,1-2H3

InChI key: InChIKey=ZZQNEJILGNNOEP-UHFFFAOYSA-N

SMILES: FC=1C=C2C(C(=NO2)C3CCN(CCC=4C(=O)N5C(=NC4C)C(C)=CC=C5)CC3)=CC1

Synonyms:

• 1,2-Benzisoxazole, 4H-pyrido[1,2-a]pyrimidin-4-one deriv.
• 3-(2-(4-(6-Fluoro-1,2-benzisoxazol-3-yl)piperidino)ethyl)-2,9-dimethyl-4H-pyrido(1,2-a)pyrimidin-4-one
• 3-[2-[4-(6-Fluoro-1,2-benzisoxazol-3-yl)-1-piperidinyl]ethyl]-2,9-dimethyl-4H-pyrido[1,2-a]pyrimidin-4-one
• 3-{2-[4-(6-fluoro-1,2-benzoxazol-3-yl)piperidin-1-yl]ethyl}-2,9-dimethyl-4H-pyrido[1,2-a]pyrimidin-4-one
• 4H-Pyrido(1,2-a)pyrimidin-4-one, 3-(2-(4-(6-fluoro-1,2-benzisoxazol-3-yl)-1-piperidinyl)ethyl)-2,9-dimethyl-
• Ocaperidona
• Ocaperidona [INN-Spanish]
• Ocaperidone [USAN:INN:BAN]
• Ocaperidonum
• Ocaperidonum [INN-Latin]
• R 79598
• Unii-26Hus7139V
• Ocaperidone
• Ocaperidone USP/EP/BP
• 5-hydroxytryptamine Receptor,Ocaperidone,inhibit,Serotonin Receptor,R 79598,Inhibitor,Dopamine Receptor,5-HT Receptor,R-79598
• R79598
• 3-(2-(4-(6-Fluorobenzo[d]isoxazol-3-yl)piperidin-1-yl)ethyl)-2,9-dimethyl-4H-pyrido[1,2-a]pyrimidin-4-one
• 3-[2-[4-(6-fluoro-1,2-benzoxazol-3-yl)piperidin-1-yl]ethyl]-2,9-dimethylpyrido[1,2-a]pyrimidin-4-one

Ocaperidone

CAS: 129029-23-8

Formula: C₂₄H₂₅FN₄O₂

Purity: >98.0%(HPLC)

Color and Shape: White to Light yellow powder to crystal

Molecular weight: 420.49

Ref: 3B-O0498

4H-Pyrido[1,2-a]pyrimidin-4-one, 3-[2-[4-(6-fluoro-1,2-benzisoxazol-3-yl)-1-piperidinyl]ethyl]-2,9-dimethyl-

CAS: 129029-23-8

Formula: C₂₄H₂₅FN₄O₂

Purity: 98%

Color and Shape: Solid

Molecular weight: 420.4793

Ref: IN-DA000YST

Ocaperidone

CAS: 129029-23-8

Ocaperidone

Purity: ≥98%

Molecular weight: 420.48g/mol

Ref: 54-BUP02789

Ocaperidone

CAS: 129029-23-8

Ocaperidona (Ocaperidone (Ocaperidona)), a very high affinity dopamine D2 antagonist.

Formula: C₂₄H₂₅FN₄O₂

Purity: 99.33%

Color and Shape: Solid

Molecular weight: 420.48

Ref: TM-T3497

Ocaperidone

Controlled Product

CAS: 129029-23-8

Applications Ocaperidone, is an effective antipsychotic agent, acting as a potent 5-HT2 and dopamine D2 antagonist.
Not a dangerous good if item is equal to or less than 1g/ml and there is less than 100g/ml in the package
References Leysen, J. E. et al.: Mol Pharmacol. 1992 Mar;41(3):494-508.; Cosi, C. et al.: Eur J Pharmacol. 2001 Dec 14;433(1):55-62.;

Formula: C₂₄H₂₅FN₄O₂

Color and Shape: Neat

Molecular weight: 420.48

Ref: TR-O234005