CAS 130800-90-7
:Sipatrigine
Description:
Sipatrigine, with the CAS number 130800-90-7, is a chemical compound that belongs to the class of substances known as sodium channel blockers. It is primarily studied for its potential therapeutic applications, particularly in the treatment of neurological disorders such as epilepsy. The compound exhibits a mechanism of action that involves the modulation of sodium ion flow across neuronal membranes, which can help stabilize neuronal excitability and reduce seizure activity. Sipatrigine is characterized by its specific molecular structure, which contributes to its pharmacological properties. In terms of solubility, it typically shows moderate solubility in organic solvents, while its solubility in water may vary. Safety and toxicity profiles are essential considerations in its development, and ongoing research aims to elucidate its efficacy and side effects in clinical settings. As with many pharmaceutical compounds, understanding its pharmacokinetics, including absorption, distribution, metabolism, and excretion, is crucial for its potential use in medical applications.
Formula:C15H16Cl3N5
InChI:InChI=1S/C15H16Cl3N5/c1-22-2-4-23(5-3-22)15-20-8-11(14(19)21-15)10-6-9(16)7-12(17)13(10)18/h6-8H,2-5H2,1H3,(H2,19,20,21)
InChI key:InChIKey=PDOCBJADCWMDGL-UHFFFAOYSA-N
SMILES:ClC1=C(C=C(Cl)C=C1Cl)C=2C(N)=NC(=NC2)N3CCN(C)CC3
Synonyms:- 2-(4-Methyl-1-piperazinyl)-5-(2,3,5-trichlorophenyl)-4-pyrimidinamine
- 2-(4-Methyl-piperazin-1-yl)-5-(2,3,5-trichloro-phenyl)-pyrimidin-4-ylamine
- 2-(4-Methylpiperazin-1-Yl)-5-(2,3,5-Trichlorophenyl)-Pyrimidin-4-Amine
- 4-Pyrimidinamine, 2-(4-methyl-1-piperazinyl)-5-(2,3,5-trichlorophenyl)-
- 619C89
- Bw 619C89
- L-Glutamic Acid, N-[4-[2-(2-Amino-4,7-Dihydro-4-8 Oxo-1H-Pyrrolo[2,3-D] Pyrimidin-5-Yl)Ethyl]Benzoyl]-, Disodium Salt, Heptahydrate
- disodium (2S)-2-[({4-[2-(2-amino-4-oxo-4,7-dihydro-1H-pyrrolo[2,3-d]pyrimidin-5-yl)ethyl]phenyl}carbonyl)amino]pentanedioate
- Sipatrigine
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Found 4 products.
4-Pyrimidinamine, 2-(4-methyl-1-piperazinyl)-5-(2,3,5-trichlorophenyl)-
CAS:Formula:C15H16Cl3N5Purity:95%Molecular weight:372.6800Sipatrigine
CAS:Sipatrigine (619C89) is an inhibitor of glutamate release, TREK ion channels, TRESK channels, sodium channels, and calcium channels.Formula:C15H16Cl3N5Purity:98.64% - 99.77%Color and Shape:SolidMolecular weight:372.68



