CAS 1310877-95-2

METHYLSTAT

Description:

Methylstat, identified by its CAS number 1310877-95-2, is a chemical compound that has garnered attention in the field of medicinal chemistry, particularly for its potential applications in cancer treatment. It is classified as a small molecule inhibitor, specifically targeting the enzyme methyltransferase, which plays a crucial role in various cellular processes, including gene expression and protein function. Methylstat's mechanism of action involves the inhibition of methylation, a post-translational modification that can influence tumor growth and progression. The compound is typically characterized by its specific molecular structure, which includes functional groups that facilitate its interaction with biological targets. In terms of physical properties, Methylstat is expected to exhibit moderate solubility in organic solvents, with stability under standard laboratory conditions. Ongoing research aims to further elucidate its pharmacokinetics, efficacy, and safety profile, making it a subject of interest for further development in therapeutic applications. As with any investigational compound, detailed studies are necessary to fully understand its biological effects and potential clinical uses.

Formula: C₂₈H₃₁N₃O₆

Synonyms:

• Methylstat >=98% (HPLC)
• MUJOCHRZXRZONW-FOCLMDBBSA-N
• (E)-methyl 4-(N-hydroxy-4-(4-((naphthalen-1-yl-carbamoyloxy)methyl)benzylamino)butylamino)-4-oxobut-2-enoate
• (2E)-4-[Hydroxy[4-[[[4-[[[(1-naphthalenylamino)carbonyl]oxy]methyl]phenyl]methyl]amino]butyl]amino]-4-oxo-2-butenoic acid methyl ester
• 2-Butenoic acid, 4-[hydroxy[4-[[[4-[[[(1-naphthalenylamino)carbonyl]oxy]methyl]phenyl]methyl]amino]butyl]amino]-4-oxo-, methyl ester, (2E)-
• JMJD Histone Demethylase Inhibitor IV, Methylstat - CAS 1310877-95-2 - Calbiochem
• METHYLSTAT
• JMJD Histone Demethylase Inhibitor IV, Methylstat

Methylstat

CAS: 1310877-95-2

Methylstat

Purity: ≥98%

Molecular weight: 505.56g/mol

Ref: 54-BUP21915

Methylstat

CAS: 1310877-95-2

Methylstat is a methyl ester prodrug of a Jumonji C domain-containing histone demethylase (JMJD) inhibitor that has favorable cell permeability.

Formula: C₂₈H₃₁N₃O₆

Purity: 98.34% - 98.34%

Color and Shape: Solid

Molecular weight: 505.56

Ref: TM-T7057

JMJD Histone Demethylase Inhibitor IV, Methylstat

CAS: 1310877-95-2

JMJD Histone Demethylase Inhibitor IV, Methylstat is a drug that inhibits the protein methyltransferase and is used to treat cancer. It has been shown to induce apoptosis in hl-60 cells by inhibiting histone proteins and altering the structure of the genome. JMJD Histone Demethylase Inhibitor IV, Methylstat also has an effect on mitochondrial membrane potential (MMP) and induces cell cycle arrest. This drug is administered orally or intravenously and is currently undergoing clinical trials for treatment of cancer.

Formula: C₂₈H₃₁N₃O₆

Purity: Min. 95%

Molecular weight: 505.56 g/mol

Ref: 3D-KCC87795