CAS 1329796-60-2

Etoperidone-d8 Hydrochloride

Description:

Etoperidone-d8 Hydrochloride is a deuterated form of etoperidone, which is an atypical antipsychotic medication primarily used in the treatment of schizophrenia and other psychiatric disorders. The "d8" designation indicates that the compound contains eight deuterium atoms, which are isotopes of hydrogen, replacing the regular hydrogen atoms in the molecular structure. This modification can enhance the stability and metabolic tracking of the compound in pharmacokinetic studies. As a hydrochloride salt, it is typically more soluble in water, facilitating its use in various formulations. The compound exhibits properties characteristic of antipsychotic agents, including dopamine receptor antagonism, which contributes to its therapeutic effects. Additionally, the deuterated version may exhibit altered pharmacodynamics and pharmacokinetics compared to its non-deuterated counterpart, making it valuable for research purposes. Safety and efficacy profiles are determined through clinical studies, and as with all pharmaceuticals, it is essential to consider potential side effects and interactions with other medications.

Formula: C₁₉H₂₉Cl₂N₅O

Synonyms:

• Etonin-d8
• Etoran-d8
• Tropene-d8
• Trazodone Impurity 54
• AxioMin-d8
• Deprecer-d8
• Staff-d8
• McN-A 2673-11-d8
• ST 1191-d8
• 2-[3-[4-(3-chlorophenyl)-2,2,3,3,5,5,6,6-octadeuteriopiperazin-1-yl]propyl]-4,5-diethyl-1,2,4-triazol-3-one:hydrochloride
• Trazodone Impurity 49
• 2-[3-[4-(3-Chlorophenyl)-1-(piperazinyl-d8)]propyl]-4,5-diethyl-2,4-dihydro-3H-1,2,4-triazol-3-one Hydrochloride
• AF 1191-d8

Etoperidone-d8 Hydrochloride

Controlled Product

CAS: 1329796-60-2

Applications Labelled Etoperidone (E933680). A psychotropic drug related structurally to trazodone. Antidepressant.
References Barcellona, S., et al.: Toxicology, 8, 87 (1977), Bertoletti, G., et al.: Clin. Med., 58, 393 (1977), Lisciani, R., et al.: Arzneim.-Forsch., 28, 417 (1978),

Formula: C₁₉H₂₁D₈Cl₂N₅O

Color and Shape: Neat

Molecular weight: 422.42

Ref: TR-E933682