CAS 133040-01-4: Eprosartan

Description: Eprosartan is an antihypertensive medication classified as an angiotensin II receptor blocker (ARB). It is primarily used to treat high blood pressure and is known for its ability to relax blood vessels, thereby reducing blood pressure and improving blood flow. The chemical formula of eprosartan is C20H24N2O4S, and it features a sulfonamide group, which contributes to its pharmacological activity. Eprosartan is characterized by its relatively high solubility in water and moderate lipophilicity, allowing for effective absorption in the gastrointestinal tract. The compound has a specific stereochemistry that is crucial for its interaction with the angiotensin II receptor. Eprosartan is typically administered orally and is often well-tolerated, with a side effect profile that may include dizziness, fatigue, and gastrointestinal disturbances. Its mechanism of action involves blocking the effects of angiotensin II, a peptide that constricts blood vessels, thus playing a significant role in the regulation of blood pressure. Overall, eprosartan is an important therapeutic agent in the management of hypertension.

Formula: C₂₃H₂₄N₂O₄S

InChI: InChI=1S/C23H24N2O4S/c1-2-3-6-21-24-14-19(12-18(23(28)29)13-20-5-4-11-30-20)25(21)15-16-7-9-17(10-8-16)22(26)27/h4-5,7-12,14H,2-3,6,13,15H2,1H3,(H,26,27)(H,28,29)/b18-12+

InChI key: InChIKey=OROAFUQRIXKEMV-LDADJPATSA-N

SMILES: O=C(O)C1=CC=C(C=C1)CN2C(=CN=C2CCCC)C=C(C(=O)O)CC=3SC=CC3

Synonyms:

• ((E)-3-[2-Butyl-1-[(4-carboxyphenyl)methyl]imidazol-5-yl]-2-(2-thienylmethyl)-2-propenoic Acid
• (E)- α-[[2-Butyl-1-[(4-carboxyphenyl)methyl]-1H-imidazol-5-y1]methylene]2-thiophenepropanoic acid
• (E)-2-Butyl-1-(p-carboxybenzyl)-α-2-thenylimidazole-5-acrylic acid
• (E)-3-[2-Butyl-1-[(4-carboxyphenyl)-methyl]imidazol-5-l]-2-(2-thienylmethyl)-2-propenoic Acid
• (αE)-α-[[2-Butyl-1-[(4-carboxyphenyl)methyl]-1H-imidazol-5-yl]methylene]-2-thiophenepropanoic acid
• 2-Thiophenepropanoic acid, α-[[2-butyl-1-[(4-carboxyphenyl)methyl]-1H-imidazol-5-yl]methylene]-, (E)-
• 2-Thiophenepropanoic acid, α-[[2-butyl-1-[(4-carboxyphenyl)methyl]-1H-imidazol-5-yl]methylene]-, (αE)-
• 4-({2-butyl-5-[(1E)-2-carboxy-3-thiophen-2-ylprop-1-en-1-yl]-1H-imidazol-1-yl}methyl)benzoic acid
• 4-({2-butyl-5-[2-carboxy-3-(thiophen-2-yl)prop-1-en-1-yl]-1H-imidazol-1-yl}methyl)benzoic acid
• Eporlosartan
• Eprosartan Mysylate
• Navixen
• Skb 108566
• Skf-108566)
• Skf-108566J
• Teveten

Eprosartan Mesylate

CAS: 133040-01-4144143-96-4

• Formula: C₂₃H₂₄N₂O₄S·CH₄O₃S
• Purity: >98.0%(T)(HPLC)
• Color and Shape: White to Almost white powder to crystal
• Molecular weight: 520.62

2-Thiophenepropanoic acid, α-[[2-butyl-1-[(4-carboxyphenyl)methyl]-1H-imidazol-5-yl]methylene]-, (αE)-

CAS: 133040-01-4

• Formula: C₂₃H₂₄N₂O₄S
• Purity: 95%
• Color and Shape: Solid
• Molecular weight: 424.5127

Eprosartan

CAS: 133040-01-4

Eprosartan is a selective AT1 receptor blocker with IC50s of 9.2 nM (rat) and 3.9 …

• Formula: C₂₃H₂₄N₂O₄S
• Purity: 100%
• Color and Shape: Solid
• Molecular weight: 424.51

Eprosartan

CAS: 133040-01-4

• Formula: C₂₃H₂₄N₂O₄S
• Molecular weight: 424.51

Eprosartan-d4

CAS: 133040-01-4

• Formula: C₂₃H₂₀N₂O₄SD₄
• Color and Shape: White To Off-White Solid
• Molecular weight: 428.55

Eprosartan

CAS: 133040-01-4

• Formula: C₂₃H₂₄N₂O₄S
• Color and Shape: Light Yellow
• Molecular weight: 424.51

Eprosartan

CAS: 133040-01-4

Please enquire for more information about Eprosartan including the price, delivery time and more detailed …

• Formula: C₂₃H₂₄N₂O₄S
• Purity: Min. 95%
• Molecular weight: 424.51 g/mol