CAS 134564-82-2

Befloxatone

Description:

Befloxatone is a chemical compound classified as a selective monoamine oxidase inhibitor (MAOI), primarily used in the treatment of depression. It functions by inhibiting the activity of the monoamine oxidase enzyme, which is responsible for the breakdown of neurotransmitters such as serotonin, norepinephrine, and dopamine in the brain. This inhibition leads to increased levels of these neurotransmitters, potentially alleviating depressive symptoms. Befloxatone is characterized by its specific action on the MAO-B isoform, which contributes to its therapeutic effects while minimizing some of the dietary restrictions typically associated with non-selective MAOIs. The compound has a relatively low solubility in water and is often administered in oral form. As with other MAOIs, it may interact with certain foods and medications, necessitating careful management to avoid hypertensive crises. Overall, befloxatone represents a targeted approach in psychopharmacology, with a focus on enhancing mood and emotional well-being through neurotransmitter modulation.

Formula: C₁₅H₁₈F₃NO₅

InChI: InChI=1S/C15H18F3NO5/c1-22-9-12-8-19(14(21)24-12)10-2-4-11(5-3-10)23-7-6-13(20)15(16,17)18/h2-5,12-13,20H,6-9H2,1H3/t12-,13-/m1/s1

InChI key: InChIKey=IALVDLPLCLFBCF-CHWSQXEVSA-N

SMILES: O=C1N(C[C@H](COC)O1)C2=CC=C(OCC[C@H](C(F)(F)F)O)C=C2

Synonyms:

• (5R)-5-(Methoxymethyl)-3-[4-[(3R)-4,4,4-trifluoro-3-hydroxybutoxy]phenyl]-2-oxazolidinone
• (5R)-5-(methoxymethyl)-3-(4-{[(3R)-4,4,4-trifluoro-3-hydroxybutyl]oxy}phenyl)-1,3-oxazolidin-2-one
• (R)-5-(Methoxymethyl)-3-(p-((R)-4,4,4-trifluoro-3-hydroxybutoxy)phenyl)-2-oxazolidinone
• 2-Oxazolidinone, 5-(methoxymethyl)-3-(4-(4,4,4-trifluoro-3-hydroxybutoxy)phenyl)-, (R,(R*,R*))-
• 2-Oxazolidinone, 5-(methoxymethyl)-3-[4-[(3R)-4,4,4-trifluoro-3-hydroxybutoxy]phenyl]-, (5R)-
• Befloxatone [INN]
• Md 370503
• Unii-4H75Pad8M3
• Befloxatone

Befloxatone

Controlled Product

CAS: 134564-82-2

Formula: C₁₅H₁₈F₃NO₅

Color and Shape: Neat

Molecular weight: 349.302

Ref: TR-B131084

Befloxatone

CAS: 134564-82-2

Befloxatone is a potent, selective and reversible inhibitor of monoamine oxidase A.

Formula: C₁₅H₁₈F₃NO₅

Color and Shape: Solid

Molecular weight: 349.3

Ref: TM-T26761