CAS: 1346574-57-9 - GSK126

Formula: C₃₁H₃₈N₆O₂

InChI: InChI=1S/C31H38N6O2/c1-6-22(5)37-18-20(3)29-25(30(38)34-17-26-19(2)13-21(4)35-31(26)39)14-24(15-27(29)37)23-7-8-28(33-16-23)36-11-9-32-10-12-36/h7-8,13-16,18,22,32H,6,9-12,17H2,1-5H3,(H,34,38)(H,35,39)/t22-/m0/s1

InChI key: InChIKey=FKSFKBQGSFSOSM-QFIPXVFZSA-N

SMILES: O=C(NCC=1C(=O)NC(=CC1C)C)C2=CC(=CC3=C2C(=CN3C(C)CC)C)C=4C=NC(=CC4)N5CCNCC5

GSK126

CAS: 1346574-57-9

• Molecular weight: 526.67g/mol

GSK126

CAS: 1346574-57-9

GSK126 (GSK2816126A) is a excellently specific EZH2 methyltransferase inhibitor ( IC50=9.9 nM).

• Formula: C₃₁H₃₈N₆O₂
• Purity: 98% - 99.67%
• Color and Shape: Solid
• Molecular weight: 526.67

GSK 126

CAS: 1346574-57-9

GSK-126 is a potent inhibitor of histone lysine methyl transferase 2, which is encoded by …

• Formula: C₃₁H₃₈N₆O₂
• Purity: Min. 95%
• Color and Shape: White To Yellow Solid
• Molecular weight: 526.30562

GSK126

CAS: 1346574-57-9

Applications GSK126 is a potent and highly selective S-adenosyl-methionine-competitive small molecule inhibitor of EZH2 methyltransferase …

• Formula: C₃₁H₃₈N₆O₂
• Color and Shape: Neat
• Molecular weight: 526.67

S)-1-(sec-butyl)-N-((4,6-diMethyl-2-oxo-1,2-dihydropyridin-3-yl)Methyl)-3-Methyl-6-(6-(piperazin-1-yl)pyridin-3-yl)-1H-indole-4-carboxaMide

CAS: 1346574-57-9

• Formula: C₃₁H₃₈N₆O₂
• Purity: 98%
• Color and Shape: Solid
• Molecular weight: 526.6724