CAS 135042-90-9

N-DescyclopropylMethyl-N-Methoxycarbonyl-6,8-dehydro-3-O-Methyl Naltrexone

Description:

N-DescyclopropylMethyl-N-Methoxycarbonyl-6,8-dehydro-3-O-Methyl Naltrexone, with CAS number 135042-90-9, is a synthetic derivative of naltrexone, which is an opioid antagonist primarily used in the treatment of opioid addiction and alcohol dependence. This compound features a complex molecular structure characterized by the presence of a methoxycarbonyl group, which enhances its pharmacological properties. The dehydro and O-methyl modifications contribute to its unique activity profile, potentially affecting its binding affinity to opioid receptors. As a result, it may exhibit altered pharmacokinetics and pharmacodynamics compared to its parent compound. The presence of the descyclopropylmethyl group suggests modifications that could influence its metabolic stability and bioavailability. While specific biological activities and therapeutic applications may require further investigation, compounds like this are often studied for their potential in pain management and addiction therapies. Safety and efficacy profiles would need to be established through rigorous clinical testing.

Formula: C₁₉H₁₉NO₅

Synonyms:

• N-DescyclopropylMethyl-N-Methoxycarbonyl-6,8-dehydro-3-O-Methyl Naltrexone
• (5α)-7,8-Didehydro-4,5-epoxy-3-Methoxy-6-oxo-Morphinan-17-carboxylic acid Methyl Ester

N-Descyclopropylmethyl-N-methoxycarbonyl-6,8-dehydro-3-O-methyl Naltrexone

Controlled Product

CAS: 135042-90-9

Applications Codeinone derivative (C635000). Used in the preparation of Naltrexone by-product.

Formula: C₁₉H₁₉NO₅

Color and Shape: Neat

Molecular weight: 341.36

Ref: TR-D291900