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CAS 135729-56-5

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Palonosetron racemic

Description:
Palonosetron racemic is a chemical compound primarily used as an antiemetic, particularly in the prevention of nausea and vomiting associated with chemotherapy and surgery. It belongs to the class of 5-HT3 receptor antagonists, which function by blocking serotonin receptors in the gastrointestinal tract and central nervous system, thereby reducing the sensation of nausea. The compound is characterized by its high affinity for the 5-HT3 receptor, which contributes to its effectiveness and prolonged action compared to other agents in the same class. Palonosetron racemic is typically administered intravenously or orally, and its pharmacokinetics indicate a relatively long half-life, allowing for less frequent dosing. The substance is generally well-tolerated, with common side effects including headache and constipation. Its racemic nature indicates that it exists as a mixture of two enantiomers, which may influence its pharmacological properties. Overall, palonosetron racemic is a significant therapeutic agent in managing chemotherapy-induced nausea and vomiting, enhancing patient comfort during cancer treatment.
Formula:C19H24N2O
InChI:InChI=1/C19H24N2O/c22-19-16-6-2-4-14-3-1-5-15(18(14)16)11-21(19)17-12-20-9-7-13(17)8-10-20/h2,4,6,13,15,17H,1,3,5,7-12H2/t15-,17-/m1/s1
SMILES:C1Cc2cccc3c2[C@H](C1)CN([C@@H]1CN2CCC1CC2)C3=O
Synonyms:
  • (3As)-2-(S)-1-Azabicyclo[2,2,2]Oct-3-Yl)-2,3,3A,4,5,6-Hexahydro-1H-Benz(D)Isoquinolin-1-One
  • Palonosteron
  • Palmatine(P) Ky-7
  • (3aS)-2-[(3S)-1-azabicyclo[2.2.2]oct-3-yl]-2,3,3a,4,5,6-hexahydro-1H-benzo[de]isoquinolin-1-one
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