CAS 138470-70-9

Mozavaptan hydrochloride

Description:

Mozavaptan hydrochloride is a chemical compound classified as a vasopressin receptor antagonist, specifically targeting the V2 receptor. It is primarily investigated for its potential therapeutic applications in conditions such as hyponatremia and heart failure. The substance appears as a white to off-white crystalline powder and is soluble in water, which facilitates its administration in clinical settings. Its molecular structure includes a specific arrangement of atoms that contributes to its biological activity, allowing it to modulate water retention in the kidneys. The compound's pharmacokinetics, including absorption, distribution, metabolism, and excretion, are crucial for determining its efficacy and safety profile. As with many pharmaceuticals, the hydrochloride salt form enhances stability and solubility. Research continues to explore its full therapeutic potential and side effects, emphasizing the importance of understanding its mechanism of action at the molecular level. Overall, Mozavaptan hydrochloride represents a significant advancement in the management of disorders related to water balance in the body.

Formula: C₂₇H₂₉N₃O₂·ClH

InChI: InChI=1S/C27H29N3O2.ClH/c1-19-9-4-5-10-22(19)26(31)28-21-16-14-20(15-17-21)27(32)30-18-8-13-24(29(2)3)23-11-6-7-12-25(23)30;/h4-7,9-12,14-17,24H,8,13,18H2,1-3H3,(H,28,31);1H

InChI key: InChIKey=MOROBKPIULFQDC-UHFFFAOYSA-N

SMILES: C(=O)(N1C=2C(C(N(C)C)CCC1)=CC=CC2)C3=CC=C(NC(=O)C4=C(C)C=CC=C4)C=C3.Cl

Synonyms:

• Mozavaptan hydrochloride
• Benzamide, N-[4-[[5-(dimethylamino)-2,3,4,5-tetrahydro-1H-1-benzazepin-1-yl]carbonyl]phenyl]-2-methyl-, hydrochloride (1:1)
• Benzamide, N-[4-[[5-(dimethylamino)-2,3,4,5-tetrahydro-1H-1-benzazepin-1-yl]carbonyl]phenyl]-2-methyl-, monohydrochloride
• 1H-1-Benzazepine, benzamide deriv.
• Benzamide, N-[4-[[5-(dimethylamino)-2,3,4,5-tetrahydro-1H-1-benzazepin-1-yl]carbonyl]phenyl]-2-methyl-, monohydrochloride, (±)-

Benzamide, N-[4-[[5-(dimethylamino)-2,3,4,5-tetrahydro-1H-1-benzazepin-1-yl]carbonyl]phenyl]-2-methyl-, hydrochloride (1:1)

CAS: 138470-70-9

Formula: C₂₇H₃₀ClN₃O₂

Purity: 98%

Color and Shape: Solid

Molecular weight: 463.9990

Ref: IN-DA00197R

Mozavaptan hydrochloride

CAS: 138470-70-9

Mozavaptan is a vasopressin receptor antagonist.

Formula: C₂₇H₃₀ClN₃O₂

Color and Shape: Solid

Molecular weight: 464

Ref: TM-T21465

Mozavaptan HCl

Controlled Product

CAS: 138470-70-9

Mozavaptan HCl is a pharmaceutical compound classified as a selective vasopressin V2 receptor antagonist, which is synthesized chemically. Mozavaptan HCl exerts its effects by inhibiting the action of the antidiuretic hormone vasopressin on renal collecting ducts. This inhibition prevents the binding of vasopressin to V2 receptors, thereby reducing water reabsorption in the kidneys.

Formula: C₂₇H₂₉N₃O₂·HCl

Purity: Min. 95%

Molecular weight: 464 g/mol

Ref: 3D-NFA47070