CAS 138742-43-5

Zankiren

Description:

Zankiren, identified by the CAS number 138742-43-5, is a chemical compound that has garnered attention in the field of medicinal chemistry, particularly for its role as a therapeutic agent. It is characterized by its specific molecular structure, which contributes to its biological activity. Zankiren functions primarily as a selective inhibitor, targeting specific enzymes or receptors within biological systems, which can lead to various pharmacological effects. The compound is often studied for its potential applications in treating certain diseases, including those related to inflammation or metabolic disorders. Its solubility, stability, and interaction with other biological molecules are critical factors that influence its efficacy and safety profile. Additionally, Zankiren's synthesis and formulation are important for its application in research and clinical settings. As with many chemical substances, understanding its mechanism of action, pharmacokinetics, and potential side effects is essential for evaluating its therapeutic potential.

Formula: C₃₅H₅₅N₅O₆S₂

InChI: InChI=1/C35H55N5O6S2/c1-25(2)18-32(41)33(42)30(20-27-12-8-5-9-13-27)37-35(44)31(21-29-22-47-24-36-29)38-34(43)28(19-26-10-6-4-7-11-26)23-48(45,46)40-16-14-39(3)15-17-40/h4,6-7,10-11,22,24-25,27-28,30-33,41-42H,5,8-9,12-21,23H2,1-3H3,(H,37,44)(H,38,43)/t28-,30+,31+,32+,33-/m1/s1

Synonyms:

• zankiren HCl
• N~2~-{(2S)-2-benzyl-3-[(4-methylpiperazin-1-yl)sulfonyl]propanoyl}-N-[(1S,2R,3S)-1-(cyclohexylmethyl)-2,3-dihydroxy-5-methylhexyl]-3-(1,3-thiazol-4-yl)alaninamide
• N~2~-{(2S)-2-benzyl-3-[(4-methylpiperazin-1-yl)sulfonyl]propanoyl}-N-[(1S,2R,3S)-1-(cyclohexylmethyl)-2,3-dihydroxy-5-methylhexyl]-3-(1,3-thiazol-4-yl)-L-alaninamide

Zankiren

CAS: 138742-43-5

Zankiren is a renin inhibitor. Zankiren can reduce blood pressure, plasma renin activity, and angiotension II.

Formula: C₃₅H₅₅N₅O₆S₂

Color and Shape: Solid

Molecular weight: 705.97

Ref: TM-T29204

Zankiren

Controlled Product

CAS: 138742-43-5

Applications Zankiren, is a drug that acts as a renin inhibitor in human. It has been also shown to be orally active in the dog and other animals.
References Wessale, J. L., et al.: American J. Hypertension, 6, 514 (1993);

Formula: C₃₅H₅₅N₅O₆S₂

Color and Shape: Neat

Molecular weight: 705.971

Ref: TR-Z148060

Zankiren

CAS: 138742-43-5

Zankiren is a peptide inhibitor of protein interactions. It has been shown to inhibit the activity of several proteins, including G-protein coupled receptors and ion channels. Zankiren is a high purity research tool that can be used for studying cell biology and pharmacology.

Formula: C₃₅H₅₅N₅O₆S₂

Purity: Min. 95%

Molecular weight: 706.00 g/mol

Ref: 3D-NFA74243