CymitQuimica logo

CAS 14009-24-6

:

Drotaverine

Description:
Drotaverine is a synthetic antispasmodic agent primarily used to relieve smooth muscle spasms in various conditions, such as gastrointestinal and biliary colic. It belongs to the class of compounds known as isoquinoline derivatives and is characterized by its ability to inhibit phosphodiesterase, leading to increased levels of cyclic adenosine monophosphate (cAMP) in smooth muscle cells. This mechanism results in muscle relaxation and alleviation of spasms. Drotaverine is typically administered orally or via injection, and it is well-absorbed in the gastrointestinal tract. The substance is known for its relatively low toxicity and side effects, making it a preferred choice in clinical settings for managing pain associated with spasmodic conditions. Its chemical structure includes a butyl group, contributing to its lipophilicity, which enhances its bioavailability. Drotaverine is often marketed under various brand names and is widely used in several countries, although its availability may vary.
Formula:C24H31NO4
InChI:InChI=1S/C24H31NO4/c1-5-26-21-10-9-17(14-22(21)27-6-2)13-20-19-16-24(29-8-4)23(28-7-3)15-18(19)11-12-25-20/h9-10,13-16,25H,5-8,11-12H2,1-4H3
InChI key:InChIKey=OMFNSKIUKYOYRG-UHFFFAOYSA-N
SMILES:C(=C1C=2C(=CC(OCC)=C(OCC)C2)CCN1)C3=CC(OCC)=C(OCC)C=C3
Synonyms:
  • (1Z)-1-(3,4-Diethoxybenzylidene)-6,7-diethoxy-1,2,3,4-tetrahydroisoquinoline
  • (1Z)-1-(3,4-diethoxybenzylidene)-6,7-diethoxy-1,2,3,4-tetrahydroisoquinolinato(4-)
  • (1Z)-1-[(3,4-diethoxyphenyl)methylidene]-6,7-diethoxy-1,2,3,4-tetrahydroisoquinoline hydrochloride
  • 1-(3,4-Diethoxybenzylidene)-6,7-diethoxy-1,2,3,4-tetrahydroisoquinoline
  • 1-(3,4-Diethoxybenzylidene)-6,7diethoxy-1,2,3,4-tetrahydroisoquinoline
  • 1-[(3,4-Diethoxyphenyl)methylene]-6,7-diethoxy-1,2,3,4-tetrahydroisoquinoline
  • 14009-24-6
  • 3′,4′,6,7-Tetraethoxy-1-benzyliden-1,2,3,4-tetrahydroisoquinoline
  • 3′,4′,6,7-Tetraethoxy-1-benzylidene-1,2,3,4-tetrahydroisoquinoline
  • DRA
  • See more synonyms
Sort by
The purity filter is not visible because current products do not have associated purity data for filtering.
Found 1 products.
  • Drotaverine
    Targetmol
    + Info

    Drotaverine

    CAS:
    Drotaverine Hydrochloride is a selective inhibitor of phosphodiesterase 4.
    Formula:C24H31NO4
    Color and Shape:Pale Yellow Powder
    Molecular weight:397.51

    Ref: TM-T19824

    25mg
    1,882.00€