CAS 140924-11-4

Piperazine, 2,6-dimethyl-1-(1-oxopropyl)-4-(3-phenyl-2-propenyl)-, [2α,4(E),6α]- (9CI)

Description:

Piperazine, 2,6-dimethyl-1-(1-oxopropyl)-4-(3-phenyl-2-propenyl)-, [2α,4(E),6α]- (9CI) is a chemical compound characterized by its piperazine core structure, which is a six-membered ring containing two nitrogen atoms. This compound features multiple substituents, including a 1-oxopropyl group and a 3-phenyl-2-propenyl moiety, contributing to its complexity and potential biological activity. The presence of the dimethyl groups at the 2 and 6 positions of the piperazine ring enhances its steric properties and may influence its interaction with biological targets. The compound's stereochemistry, indicated by the [2α,4(E),6α] notation, suggests specific spatial arrangements that can affect its pharmacological profile. Piperazine derivatives are often studied for their potential therapeutic applications, including in the fields of psychiatry and neurology, due to their ability to interact with neurotransmitter systems. However, detailed studies on the specific biological activity and safety profile of this compound would be necessary to fully understand its potential uses.

Formula: C₁₈H₂₆N₂O

Synonyms:

• AP-238
• Piperazine, 2,6-dimethyl-1-(1-oxopropyl)-4-(3-phenyl-2-propenyl)-, [2α,4(E),6α]- (9CI)

AP-238

CAS: 140924-11-4

AP-238 is a novel synthetic opioid (NSO) that acts as an agonist for the μ-opioid receptor (MOR), with an EC50 of 248 nM. Additionally, AP-238 exhibits analgesic properties.

Formula: C₁₈H₂₆N₂O

Color and Shape: Solid

Molecular weight: 286.41

Ref: TM-T203057