CAS 1421866-48-9

Apimostinel

Description:

Apimostinel, with the CAS number 1421866-48-9, is a chemical compound that has garnered attention in the field of pharmacology, particularly for its potential therapeutic applications. It is classified as a small molecule and is known to act as a selective modulator of the immune system. Apimostinel has been investigated for its role in enhancing immune responses, making it a candidate for treating various autoimmune diseases and conditions where immune modulation is beneficial. The compound exhibits a unique mechanism of action that distinguishes it from traditional immunosuppressants, potentially offering a more targeted approach with fewer side effects. Its chemical structure includes specific functional groups that contribute to its biological activity, although detailed structural information is typically found in specialized databases or scientific literature. As research continues, the full spectrum of its pharmacokinetics, efficacy, and safety profile is being evaluated to determine its viability in clinical settings.

Formula: C₂₅H₃₇N₅O₆

Synonyms:

• (2S,3S)-N-((2S,3R)-1-amino-3-hydroxy-1-oxobutan-2-yl)-1-((S)-1-((2S,3R)-2-amino-3-hydroxybutanoyl)pyrrolidine-2-carbonyl)-3-benzylpyrrolidine-2-carbox
• (R)-1-(L-threonyl-L-prolyl)-N-((2S,3R)-1-amino-3-hydroxy-1-oxobutan-2-yl)-2-benzylpyrrolidine-2-carboxamide
• AGN-241660
• NRX-1074
• Apimostinel
• L-Threoninamide, L-threonyl-L-prolyl-2-(phenylmethyl)-L-prolyl-
• (2S,3S)-N-((2S,3R)-1-amino-3-hydroxy-1-oxobutan-2-yl)-1-((S)-1-((2S,3R)-2-amino-3-hydroxybutanoyl)pyrrolidine-2-carbonyl)-3-benzylpyrrolidine-2-carboxamide

Apimostinel

CAS: 1421866-48-9

Apimostinel (NRX-1074; AGN-241660) is a partial agonist of NMDA receptor.

Formula: C₂₅H₃₇N₅O₆

Color and Shape: Solid

Molecular weight: 503.59

Ref: TM-T14306

Apimostinel

CAS: 1421866-48-9

Apimostinel is a peptide-based therapeutic agent, which is derived from a modification of endogenous neuropeptides. It is designed to selectively modulate the NMDA receptor, a subtype of glutamate receptor, which plays a crucial role in synaptic plasticity and neural communication. Apimostinel functions as a partial agonist of the glycine site on the NMDA receptor. This mechanism supports synaptic strength and plasticity without the excessive activation associated with excitotoxicity, thereby providing potential neuroprotective effects.

Formula: C₂₅H₃₇N₅O₆

Purity: Min. 95%

Molecular weight: 503.6 g/mol

Ref: 3D-WGC86648