CAS 142227-51-8: 5'-HYDROXYPHENYL CARVEDILOL

Description: 5'-Hydroxyphenyl carvedilol is a derivative of carvedilol, which is a non-selective beta-blocker and alpha-1 blocker used primarily in the treatment of hypertension and heart failure. This compound features a hydroxyl group at the 5' position of the phenyl ring, which may influence its pharmacological properties and interactions. The presence of the hydroxyl group can enhance solubility and potentially alter the compound's binding affinity to adrenergic receptors. As a chemical entity, it is characterized by its molecular structure, which includes a chiral center, contributing to its stereoisomerism. The compound is typically studied for its potential therapeutic effects, including antioxidant properties and its role in cardiovascular health. Its CAS number, 142227-51-8, allows for precise identification in chemical databases. Overall, 5'-hydroxyphenyl carvedilol represents an interesting area of research in medicinal chemistry, particularly in the development of more effective cardiovascular agents with improved safety profiles.

Formula: C₂₄H₂₆N₂O₅

InChI: InChI=1/C24H26N2O5/c1-29-21-10-9-16(27)13-23(21)30-12-11-25-14-17(28)15-31-22-8-4-7-20-24(22)18-5-2-3-6-19(18)26-20/h2-10,13,17,25-28H,11-12,14-15H2,1H3

Synonyms:

• 3-[2-[[3-(9H-Carbazol-4-yloxy)-2-hydroxypropyl]amino]ethoxy]-4-methoxyphenol
• 5-Hydroxycarvedilol
• Bm 140830

Phenol, 3-[2-[[3-(9H-carbazol-4-yloxy)-2-hydroxypropyl]amino]ethoxy]-4-methoxy-

CAS: 142227-51-8

• Formula: C₂₄H₂₆N₂O₅
• Color and Shape: Solid
• Molecular weight: 422.4736

5'-Hydroxyphenyl Carvedilol

CAS: 142227-51-8

• Formula: C₂₄H₂₆N₂O₅
• Color and Shape: Off-White Solid
• Molecular weight: 422.48

5’-Hydroxyphenyl Carvedilol

CAS: 142227-51-8

Applications A metabolite of Carvedilol (C184625). It is used in the treatment of hypertension. References …

• Formula: C₂₄H₂₆N₂O₅
• Color and Shape: Neat
• Molecular weight: 422.47

5'-Hydroxyphenyl carvedilol

CAS: 142227-51-8

5'-Hydroxyphenyl carvedilol is a metabolite of enalaprilat, which is an angiotensin-converting enzyme (ACE) inhibitor. It …

• Formula: C₂₄H₂₆N₂O₅
• Purity: Min. 95%
• Molecular weight: 422.47 g/mol