CAS 142344-87-4

GP 531

Description:

GP 531, with the CAS number 142344-87-4, is a chemical compound that belongs to a class of substances known for their potential therapeutic applications, particularly in the field of neuroscience. It is recognized as a selective antagonist of certain receptors, which may influence various physiological processes. The compound is often studied for its effects on neurotransmitter systems, particularly those related to mood and cognition. GP 531's structure typically includes functional groups that contribute to its biological activity, making it a subject of interest in pharmacological research. While specific characteristics such as solubility, stability, and reactivity can vary, GP 531 is generally evaluated for its efficacy and safety in preclinical and clinical studies. As with many compounds in this category, understanding its mechanism of action and potential side effects is crucial for its development as a therapeutic agent. Further research is necessary to fully elucidate its properties and applications in medicine.

Formula: C₁₆H₂₁N₅O₄

InChI: InChI=1/C16H21N5O4/c17-14-11(15(18)24)20-8-21(14)16-13(23)12(22)10(25-16)7-19-6-9-4-2-1-3-5-9/h1-5,8,10,12-13,16,19,22-23H,6-7,17H2,(H2,18,24)/t10-,12-,13-,16-/m1/s1

SMILES: c1ccc(cc1)CNC[C@@H]1[C@H]([C@H]([C@H](n2cnc(c2N)C(=N)O)O1)O)O

Synonyms:

• 5-Amino-1-beta-D-(5'-benzylamino-5'-deoxyribofuranosyl)imidazole-4-carboxamide
• 1H-Imidazole-4-carboxamide, 5-amino-1-(5-deoxy-5-((phenylmethyl)amino)-beta-D-ribofuranosyl)-
• 5-amino-1-[5-(benzylamino)-5-deoxy-beta-D-ribofuranosyl]-1H-imidazole-4-carboxamide
• GP-531
• 1H-Imidazole-4-carboxamide, 5-amino-1-[5-deoxy-5-[(phenylmethyl)amino]-β-D-ribofuranosyl]-
• GP531,GP-531

GP531

CAS: 142344-87-4

GP531 is an analog of adenosine that has been proven to act as an agonist at A1 receptors. It has been shown to reduce the incidence of cardiac arrhythmias in an experimental model of myocardial infarction. GP531 binds to the A1 receptor with a high affinity, and its effect on cardiac arrhythmia is mediated through the activation of adenosine receptors in cardiac tissue. This drug also has effects on neutrophils and amines, but does not have any antiviral activity. GP531 does not affect plasma levels of endogenous adenosine, which may be due to its low affinity for A2 receptors.

Formula: C₁₆H₂₁N₅O₄

Purity: Min. 95%

Molecular weight: 347.37 g/mol

Ref: 3D-SFA34487

GP531

CAS: 142344-87-4

GP531, a second-gen adenosine regulator, is inactive at rest but boosts adenosine in ischemia.

Formula: C₁₆H₂₁N₅O₄

Color and Shape: Solid

Molecular weight: 347.37

Ref: TM-T13713