CAS 142872-84-2

RX871024

CAS: 142872-84-2

RX871024 is a drug that targets β-cells and has been shown to be effective in reducing the number of β-cells in diabetic patients. It also reduces the levels of epoxyeicosatrienoic acids, which are cytotoxic to β-cells. RX871024 inhibits cytosolic calcium ion levels by binding to the cytosol and blocking intracellular targets such as diacylglycerol and beta-cell apoptosis. The drug also increases phosphorylation of amp-activated protein kinase, which is necessary for glucose transport into the cell. RX871024 may have potential as a treatment for diabetes mellitus type 2 because it antagonizes pge2 in wild-type mice.

Formula: C₁₇H₁₆ClN₃

Purity: Min. 95%

Molecular weight: 297.8 g/mol

Ref: 3D-SFA87284