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CAS 144034-80-0

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Rizatriptan

Description:
Rizatriptan is a selective serotonin receptor agonist primarily used in the treatment of acute migraine attacks. It belongs to the triptan class of medications, which are designed to alleviate migraine symptoms by targeting serotonin receptors in the brain, specifically the 5-HT_1B and 5-HT_1D subtypes. The chemical formula of rizatriptan is C_17H_19N_3O_2, and it has a molecular weight of approximately 295.35 g/mol. Rizatriptan is typically administered orally and is known for its rapid onset of action, making it effective in providing relief from migraine symptoms. It is characterized by its relatively high solubility in water and moderate lipophilicity, which influences its pharmacokinetic properties. Common side effects may include dizziness, fatigue, and nausea, while contraindications include cardiovascular conditions due to the potential for vasoconstriction. Overall, rizatriptan is a valuable option in migraine management, offering targeted relief for individuals suffering from this debilitating condition.
Formula:C15H19N5
InChI:InChI=1S/C15H19N5/c1-19(2)6-5-13-8-17-15-4-3-12(7-14(13)15)9-20-11-16-10-18-20/h3-4,7-8,10-11,17H,5-6,9H2,1-2H3
InChI key:InChIKey=ULFRLSNUDGIQQP-UHFFFAOYSA-N
SMILES:C(CN(C)C)C=1C=2C(NC1)=CC=C(CN3C=NC=N3)C2
Synonyms:
  • 1H-Indole-3-ethanamine, N,N-dimethyl-5-(1H-1,2,4-triazol-1-ylmethyl)-
  • 2-(5-((1H-1,2,4-Triazol-1-yl)methyl)-1H-indol-3-yl)-N,N-dimethylethanamine
  • 3-[2-(Dimethylamino)ethyl]-5-(1H-1,2,4-triazol-1-ylmethyl)indole
  • MK 462 free base
  • N,N-Dimethyl-2-[5-(1,2,4-Triazol-1-Ylmethyl)-1H-Indol-3-Yl]Ethanamine
  • N,N-Dimethyl-2-[5-(1H-1,2,4-triazol-1-ylmethyl)-1H-indol-3-yl]ethylamine
  • N,N-Dimethyl-5-(1H-1,2,4-Triazol-1-Ylmethyl)-1H-Indole-3-Ethanamine
  • N,N-dimethyl-2-[5-(1H-1,2,4-triazol-1-ylmethyl)-1H-indol-3-yl]ethanamine benzoate (1:1)
  • Risatriptan
  • Rizatriptan
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Found 3 products.