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CAS 144034-84-4

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DESMETHYL RIZATRIPTAN

Description:
Desmethyl rizatriptan, with the CAS number 144034-84-4, is a chemical compound that serves as a metabolite of rizatriptan, a medication commonly used to treat migraines. It belongs to the triptan class of drugs, which are characterized by their selective agonism of serotonin receptors, particularly the 5-HT_1B and 5-HT_1D subtypes. This compound is typically a white to off-white solid and is soluble in organic solvents, reflecting its moderate lipophilicity. Desmethyl rizatriptan exhibits pharmacological properties similar to those of its parent compound, contributing to vasoconstriction of cranial blood vessels and alleviating migraine symptoms. Its metabolic pathway involves the demethylation of rizatriptan, and understanding its characteristics is crucial for evaluating its efficacy and safety profile in clinical settings. As with many pharmacologically active substances, it is essential to consider its potential side effects and interactions with other medications.
Formula:C14H17N5
InChI:InChI=1/C14H17N5/c1-15-5-4-12-7-17-14-3-2-11(6-13(12)14)8-19-10-16-9-18-19/h2-3,6-7,9-10,15,17H,4-5,8H2,1H3
SMILES:CNCCc1c[nH]c2ccc(cc12)Cn1cncn1
Synonyms:
  • N10-Monodesmethyl Rizatriptan
  • N-Methyl-5-(1H-1,2,4-triazol-1-ylmethyl)-1H-indole-3-ethanamine
  • N-methyl-2-[5-(1H-1,2,4-triazol-1-ylmethyl)-1H-indol-3-yl]ethanamine
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