CAS 1443331-82-5

Enzalutamide-d3

CAS: 1443331-82-5

Formula: C₂₁H₁₃D₃F₄N₄O₂S

Color and Shape: White To Off-White Solid

Molecular weight: 467.46

Ref: 4Z-E-068004

Enzalutamide-d3

CAS: 1443331-82-5

Enzalutamide D3 is a deuterium labeled Enzalutamide . Enzalutamide is an androgen receptor (AR) antagonist with an IC50 of 36 nM in LNCaP prostate cells.

Formula: C₂₁H₁₆F₄N₄O₂S

Color and Shape: Solid

Molecular weight: 467.45

Ref: TM-T11208

MDV 3100-d3

Controlled Product

CAS: 1443331-82-5

Applications Labelled MDV 3100. MDV 3100 is an androgen-receptor antagonist that blocks androgens from binding to the androgen receptor and prevents nuclear translocation and co-activator recruitment of the ligand-receptor complex. MDV 3100 has also been shown to induce tumor cell apoptosis, and has no agonist activity. MDV 3100 is a candidate for the treatment of castration-resistant prostate cancer.
References Scher, H.I. et al.: Lancet, 375, 1437 (2010); Bellmunt, J. et al.: Ther. Adv. Med. Oncol., 2, 189 (2010); Ryan, C.J. et al.: J. Clin. Oncol., 29, 3651 (2011);

Formula: C₂₁H₁₃D₃F₄N₄O₂S

Color and Shape: Neat

Molecular weight: 467.45

Ref: TR-M199802

MDV 3100-d3

CAS: 1443331-82-5

MDV 3100-d3 is a research tool and activator of the Ligand Receptor Complex. It is used in Cell Biology to study protein interactions and the pharmacology of peptides, as well as in molecular biology and biochemistry. MDV 3100-d3 binds to ion channels and can be used to inhibit their function. This inhibitor has been shown to have high purity, which makes it a valuable research tool for studying protein interactions and the pharmacology of peptides.

Formula: C₂₁H₁₃D₃F₄N₄O₂S

Purity: Min. 95%

Molecular weight: 467.5 g/mol

Ref: 3D-THC33182