CAS 145158-71-0

Tegaserod

Description:

Tegaserod is a selective serotonin receptor agonist primarily used as a medication for the treatment of irritable bowel syndrome (IBS) and chronic constipation. It acts mainly on the 5-HT4 receptor, promoting gastrointestinal motility and enhancing peristalsis. The substance is characterized by its molecular formula, which includes carbon, hydrogen, nitrogen, and oxygen atoms, reflecting its organic nature. Tegaserod is typically administered orally and has a relatively short half-life, necessitating multiple doses throughout the day for effective management of symptoms. Its pharmacological profile includes potential side effects such as gastrointestinal discomfort, headache, and cardiovascular risks, which have led to its restricted use in certain populations. The compound is classified as a prescription medication and is not recommended for patients with a history of cardiovascular disease. Overall, Tegaserod represents a targeted approach to managing specific gastrointestinal disorders, highlighting the importance of receptor selectivity in drug design and therapeutic efficacy.

Formula: C₁₆H₂₃N₅O

InChI: InChI=1S/C16H23N5O/c1-3-4-5-8-18-16(17)21-20-11-12-10-19-15-7-6-13(22-2)9-14(12)15/h6-7,9-11,19H,3-5,8H2,1-2H3,(H3,17,18,21)

InChI key: InChIKey=IKBKZGMPCYNSLU-UHFFFAOYSA-N

SMILES: C(=NNC(NCCCCC)=N)C=1C=2C(NC1)=CC=C(OC)C2

Synonyms:

• (2E)-2-[(5-Methoxy-1H-indol-3-yl)methylene]-N-pentylhydrazinecarboximidamide
• (2E)-2-[(5-methoxy-1H-indol-3-yl)methylidene]-N'-pentylhydrazinecarboximidamide
• (2E)-2-[(5-methoxy-1H-indol-3-yl)methylidene]-N-pentylhydrazinecarboximidamide (2E)-but-2-enedioate (1:1)
• 145158-71-0
• 2-[(5-Methoxy-1H-indol-3-yl)methylene]-N-pentylhydrazinecarboximidamide
• Hydrazinecarboximidamide, 2-[(5-methoxy-1H-indol-3-yl)methylene]-N-pentyl-
• Zelmac
• hydrazinecarboximidamide, 2-[(5-methoxy-1H-indol-3-yl)methylene]-N-pentyl-, (2E)-
• Tegaserod
• Tegaserod

Hydrazinecarboximidamide, 2-[(5-methoxy-1H-indol-3-yl)methylene]-N-pentyl-

CAS: 145158-71-0

Formula: C₁₆H₂₃N₅O

Purity: 95%

Color and Shape: Solid

Molecular weight: 301.3867

Ref: IN-DA001KMZ

Tegaserod

CAS: 145158-71-0

Tegaserod

Purity: ≥98%

Molecular weight: 301.39g/mol

Ref: 54-BUP21518

Tegaserod

CAS: 145158-71-0

Tegaserod is a 5-HT4R agonist and 5-HT2B receptor antagonist with antitumor activity used in the treatment of irritable bowel syndrome (IBS).

Formula: C₁₆H₂₃N₅O

Purity: 99.20% - 99.89%

Color and Shape: Solid

Molecular weight: 301.39

Ref: TM-T60680

Tegaserod-d9

Controlled Product

CAS: 145158-71-0

Formula: C₁₆D₉H₁₄N₅O

Color and Shape: Neat

Molecular weight: 280.377

Ref: TR-T234890

Tegaserod

CAS: 145158-71-0

5-HT4 serotonin receptor antagonist; used to treat irritable bowel syndrome

Formula: C₁₆H₂₃N₅O

Purity: Min. 95%

Molecular weight: 301.39 g/mol

Ref: 3D-FT39316