CAS 147084-10-4

Alcaftadine

Description:

Alcaftadine is an antihistamine compound primarily used in ophthalmic formulations for the treatment of allergic conjunctivitis. It functions as a selective H1 receptor antagonist, helping to alleviate symptoms such as itching, redness, and swelling of the eyes caused by allergens. The chemical structure of Alcaftadine includes a piperidine ring, which contributes to its pharmacological activity. It is characterized by its relatively low solubility in water, which is typical for many antihistamines, and it is often formulated in eye drops for localized action. Alcaftadine has a rapid onset of action, providing relief from allergic symptoms shortly after administration. Additionally, it is known for its minimal sedative effects compared to first-generation antihistamines, making it a preferred choice for patients who require allergy relief without significant drowsiness. As with any medication, potential side effects may include local irritation or discomfort upon application, but these are generally mild and transient. Overall, Alcaftadine represents a valuable option in the management of allergic eye conditions.

Formula: C₁₉H₂₁N₃O

InChI: InChI=1S/C19H21N3O/c1-21-9-6-15(7-10-21)18-17-5-3-2-4-14(17)8-11-22-16(13-23)12-20-19(18)22/h2-5,12-13H,6-11H2,1H3

InChI key: InChIKey=MWTBKTRZPHJQLH-UHFFFAOYSA-N

SMILES: C(=O)C=1N2C(C(C=3C(CC2)=CC=CC3)=C4CCN(C)CC4)=NC1

Synonyms:

• 11-(1-Methylpiperidin-4-ylidene)-5,6-dihydroimidazo[2,1-b][3]benzazepine-3-carbaldehyde
• 5H-Imidazo(2,1-b)(3)benzazepine-3-carboxaldehyde, 6,11-dihydro-11-(1-methyl-4- piperidinylidene)-
• 6,11-Dihydro-11-(1-methyl-4-piperidinylidene)-5H-imidazo[2,1-b][3]benzazepine-3-carboxaldehyde
• Lastacaft
• R 89674
• Unii-7Z8O94Ecsx
• Alcaftadine

Alcaftadine

CAS: 147084-10-4

Formula: C₁₉H₂₁N₃O

Purity: 98%

Color and Shape: Solid

Molecular weight: 307.3895

Ref: IN-DA019FUT

Alcaftadine

CAS: 147084-10-4

Alcaftadine

Purity: ≥98%

Molecular weight: 307.39g/mol

Ref: 54-BUP13636

Alcaftadine

CAS: 147084-10-4

Formula: C₁₉H₂₁N₃O

Color and Shape: Pale Yellow Solid

Molecular weight: 307.40

Ref: 4Z-A-199001

Alcaftadine

CAS: 147084-10-4

Formula: C₁₉H₂₁N₃O

Purity: >98.0%(GC)

Color and Shape: White to Yellow to Orange powder to crystal

Molecular weight: 307.40

Ref: 3B-A3237

Alcaftadine-13C-D3

CAS: 147084-10-4

Formula: C₁₉H₁₈N₃OD₃

Molecular weight: 311.41

Ref: 4Z-A-199002

Alcaftadine

CAS: 147084-10-4

Alcaftadine (Lastacaft) is an H1 histamine receptor antagonist indicated for the prevention of itching associated with allergic conjunctivitis.

Formula: C₁₉H₂₁N₃O

Purity: 98% - 98.65%

Color and Shape: Solid

Molecular weight: 307.39

Ref: TM-T2533

Alcaftadine Acid N-Demethylated

Controlled Product

CAS: 147084-10-4

Formula: C₁₈H₁₉N₃O₂

Color and Shape: Neat

Molecular weight: 309.362

Ref: TR-A514545

Alcaftadine-N-demethylated

Controlled Product

CAS: 147084-10-4

Formula: C₁₈H₁₉N₃O

Color and Shape: Neat

Molecular weight: 293.363

Ref: TR-A514543