CAS 154674-81-4

Ac-Tyr-Val-Ala-Asp-2,6-dimethylbenzoyloxymethylketone

Description:

Ac-Tyr-Val-Ala-Asp-2,6-dimethylbenzoyloxymethylketone, identified by its CAS number 154674-81-4, is a synthetic compound that belongs to a class of molecules known as peptide derivatives. This substance features a sequence of amino acids, specifically tyrosine (Tyr), valine (Val), alanine (Ala), and aspartic acid (Asp), which are linked together to form a peptide chain. The presence of the 2,6-dimethylbenzoyloxymethylketone moiety suggests that it possesses a ketone functional group, which may contribute to its reactivity and potential applications in biochemical research or drug development. The compound's structure indicates that it may exhibit specific biological activities, possibly related to its peptide components, which can influence cellular processes. Additionally, the presence of the acetyl group (Ac) at the N-terminus may enhance its stability and bioavailability. Overall, this compound is of interest in the fields of medicinal chemistry and biochemistry, particularly for its potential roles in therapeutic applications or as a research tool in studying peptide interactions.

Formula: C₃₃H₄₂N₄O₁₀

Synonyms:

• Ac-Yvad-2,6-Dimethylbenzoyloxymethylketone

Ac-YVAD-AOM

CAS: 154674-81-4

Ac-YVAD-AOM

Purity: ≥98%

Molecular weight: 654.71g/mol

Ref: 54-BUP01395

Ac-Tyr-Val-Ala-Asp-2,6-dimethylbenzoyloxymethylketone

CAS: 154674-81-4

Ac-Tyr-Val-Ala-Asp-2,6-dimethylbenzoyloxymethylketone is a potent transcriptional regulator that can be used to treat breast cancer. Ac-Tyr-Val-Ala-Asp-2,6-dimethylbenzoyloxymethylketone binds to estrogen receptor and prevents the binding of estrogen to its receptor. This leads to the death of cancer cells by inhibiting the function of bcl family proteins. Acetylation of this compound at C8, C10, and C17 positions increases its potency in vivo. In addition, Acetylated TAVADM can inhibit pancreatic cancer cell growth by activating signal transducer and activator of transcription 3 (STAT3) and inhibiting the activity of bcl family proteins such as BCL2 and BCLXL. Acetylated TAVADM has also been shown to have antiapoptotic

Formula: C₃₃H₄₂N₄O₁₀

Purity: Min. 95%

Molecular weight: 654.71 g/mol

Ref: 3D-FA111062

Ac-YVAD-AOM

CAS: 154674-81-4

Ac-YVAD-AOM is a selective and potent caspase-1 inhibitor showing antitumor activity and potential analgesic activity.

Formula: C₃₃H₄₂N₄O₁₀

Purity: 98%

Color and Shape: Solid

Molecular weight: 654.71

Ref: TM-T78631