CAS 157263-00-8

MK 996

Description:

MK 996, also known by its CAS number 157263-00-8, is a chemical compound that belongs to the class of selective serotonin reuptake inhibitors (SSRIs). It is primarily investigated for its potential therapeutic effects in treating various mood disorders, including depression and anxiety. The compound functions by modulating serotonin levels in the brain, which can help improve mood and emotional balance. MK 996 exhibits a specific mechanism of action that targets serotonin transporters, thereby enhancing serotonin availability in synaptic clefts. In terms of physical properties, MK 996 is typically characterized by its molecular structure, which includes specific functional groups that contribute to its pharmacological activity. Safety and toxicity profiles are essential considerations in its development, and ongoing research aims to elucidate its efficacy and side effects in clinical settings. As with any pharmaceutical compound, regulatory approval and thorough clinical testing are crucial steps before it can be widely used in medical practice.

Formula: C₃₀H₂₈N₄O₃S

InChI: InChI=1/C30H28N4O3S/c1-4-27-32-28-20(2)18-21(3)31-29(28)34(27)19-22-14-16-23(17-15-22)25-12-8-9-13-26(25)38(36,37)33-30(35)24-10-6-5-7-11-24/h5-18H,4,19H2,1-3H3,(H,33,35)

SMILES: CCc1nc2c(C)cc(C)nc2n1Cc1ccc(cc1)c1ccccc1S(=O)(=O)N=C(c1ccccc1)O

Synonyms:

• 3-((2'-(Benzoylaminosulfonyl)biphenyl-4-yl)methyl)-2-ethyl-5,7-dimethyl-3H-imidazo(4,5-b)pyridine
• L 159282
• Benzamide, N-((4'-((2-ethyl-5,7-dimethyl-3H-imidazo(4,5-b)pyridin-3-yl)methyl)(1,1'-biphenyl)-2-yl)sulfonyl)-
• N-({4'-[(2-ethyl-5,7-dimethyl-3H-imidazo[4,5-b]pyridin-3-yl)methyl]biphenyl-2-yl}sulfonyl)benzamide
• MK-996

N-((4-((2-Ethyl-5,7-dimethyl-3H-imidazo[4,5-b]pyridin-3-yl)methyl)-[1,1'-biphenyl]-2-yl)sulfonyl)benzamide

CAS: 157263-00-8

Formula: C₃₀H₂₈N₄O₃S

Molecular weight: 524.6333

Ref: IN-DA001PC6

3-((2'-(Benzoylaminosulfonyl)biphenyl-4-yl)methyl)-2-ethyl-5,7-dimethyl-3H-imidazo(4,5-B)pyridine

CAS: 157263-00-8

3-((2'-(Benzoylaminosulfonyl)biphenyl-4-yl)methyl)-2-ethyl-5,7-dimethyl-3H-imidazo(4,5-B)pyridine is an at1 receptor antagonist that has been shown to be an orally active drug with a pressor effect. This compound inhibits the binding of neurokinin 1 to its receptor, leading to vasodilation and reduced blood pressure. 3-(2'-benzoylaminosulfonyl)biphenyl-4-ylmethyl)-2-ethyl-5,7-dimethyl-3H-[imidazo(4,5,-B)]pyridine has also been shown to have antihypertensive activity in animal models. The pharmacokinetics of 3-(2'-benzoylaminosulfonyl)biphenyl--4--ylmethyl)-2--ethyl--5,7--dim

Formula: C₃₀H₂₈N₄O₃S

Purity: Min. 95%

Molecular weight: 524.6 g/mol

Ref: 3D-HGA26300

L-159282

CAS: 157263-00-8

L-159282 is an orally active and nonpeptide angiotensin II receptor antagonist. It also has anti-hypertensive activity.

Formula: C₃₀H₂₈N₄O₃S

Purity: 98%

Color and Shape: Solid

Molecular weight: 524.63

Ref: TM-T15680