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CAS 1588870-36-3

:

Tankyrase-IN-2

Description:
Tankyrase-IN-2, identified by its CAS number 1588870-36-3, is a small molecule inhibitor specifically targeting tankyrase enzymes, which are part of the poly(ADP-ribose) polymerase (PARP) family. These enzymes play a crucial role in various cellular processes, including the regulation of Wnt signaling and telomere maintenance. The inhibition of tankyrases has garnered interest in cancer research, particularly for its potential to disrupt tumor growth and enhance the efficacy of certain cancer therapies. Tankyrase-IN-2 is characterized by its ability to selectively bind to the tankyrase active site, thereby preventing the poly(ADP-ribosyl)ation of target proteins. This compound is typically studied in the context of its pharmacological properties, including its potency, selectivity, and bioavailability. Additionally, its chemical structure may include specific functional groups that contribute to its inhibitory activity. Overall, Tankyrase-IN-2 represents a promising avenue for therapeutic development in oncology, particularly in cancers where tankyrase activity is dysregulated.
Formula:C17H14F2N2O2
Synonyms:
  • TankyraseIN2,Tankyrase IN 2
  • Tankyrase-IN-2
  • 4(3H)-Quinazolinone, 6,8-difluoro-2-[4-(1-hydroxy-1-methylethyl)phenyl]-
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Found 2 products.
  • Tankyrase-in-2
    Biosynth
    + Info

    Tankyrase-in-2

    CAS:
    <p>Tankyrase-in-2 is a protein that regulates the translation of mRNA by binding to the 3'UTR of mRNA. Tankyrase-in-2 is a potent inhibitor of tankyrases, which are enzymes that regulate the translation of mRNA by binding to the 3'UTR of mRNA. Tankyrase-in-2 is a high purity, recombinant antibody fragment and can be used as a research tool in various fields such as pharmacology, protein interactions, and cell biology. This product has CAS No. 1588870-36-3 and peptides sequence CAGAASKGGLESGGGLGSLD.<br>Tankyrase-in-2 can be used as an inhibitor for tankyrases.</p>
    Formula:C17H14F2N2O2
    Purity:Min. 95%
    Molecular weight:316.3 g/mol

    Ref: 3D-NNC87036

    5mg
    1,135.00€
    10mg
    1,579.00€
    25mg
    2,883.00€
    50mg
    4,613.00€
  • Tankyrase-IN-2
    Targetmol
    + Info

    Tankyrase-IN-2

    CAS:
    Tankyrase-IN-2 is a selective, potent and orally active inhibitor of tankyrase with IC50s of 10, 7, and 710 nM for TNKS1, TNKS2 as well as PARP1, respectively
    Formula:C17H14F2N2O2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:316.3

    Ref: TM-T13078

    25mg
    1,330.00€
    50mg
    1,730.00€
    100mg
    2,375.00€