CAS 1598383-41-5

Epz011989 trifluoroacetate

CAS: 1598383-41-5

EPZ011989 trifluoroacetate is a small molecule inhibitor, specifically targeting the EZH2 methyltransferase. This enzyme is a part of the Polycomb-group proteins, originating from the human chromatin-modifying system, which plays a vital role in epigenetic gene regulation. The mode of action involves the inhibition of methyltransferase activity, reducing the trimethylation of histone H3 on lysine 27 (H3K27me3), a modification linked to the repression of gene transcription.

Formula: C₃₇H₅₂F₃N₅O₆

Purity: Min. 95%

Molecular weight: 719.8 g/mol

Ref: 3D-YNC38341