CAS 16320-04-0: Gestrinone
Description:Gestrinone is a synthetic steroid with progestational and antiestrogenic properties, primarily used in the treatment of endometriosis and other gynecological disorders. It is classified as a synthetic derivative of testosterone and exhibits a unique mechanism of action by modulating hormonal pathways. Gestrinone functions by inhibiting the secretion of gonadotropins, which in turn reduces estrogen levels, thereby alleviating symptoms associated with estrogen-dependent conditions. The compound is typically administered orally and is characterized by its lipophilic nature, allowing for effective absorption and distribution in the body. Its chemical structure includes a cyclopentene ring, contributing to its biological activity. While Gestrinone is effective in managing certain medical conditions, it may also have side effects, including hormonal imbalances and potential impacts on liver function. As with any medication, its use should be closely monitored by healthcare professionals to ensure safety and efficacy. Overall, Gestrinone represents a significant option in the pharmacological management of specific reproductive health issues.
Formula:C21H24O2
InChI:InChI=1S/C21H24O2/c1-3-20-11-9-17-16-8-6-15(22)13-14(16)5-7-18(17)19(20)10-12-21(20,23)4-2/h2,9,11,13,18-19,23H,3,5-8,10,12H2,1H3/t18-,19+,20+,21+/m1/s1
InChI key:InChIKey=BJJXHLWLUDYTGC-ANULTFPQSA-N
SMILES:O=C1C=C2C(=C3C=CC4(CC)C(CCC4(O)C#C)C3CC2)CC1
- Synonyms:
- (17α)-13-Ethyl-17-hydroxy-18,19-dinorpregna-4,9,11-trien-20-yn-3-one
- (8S,13S,14S,17R)-13-ethyl-17-ethynyl-17-hydroxy-1,2,6,7,8,13,14,15,16,17-decahydro-3H-cyclopenta[a]phenanthren-3-one (non-preferred name)
- 13-Ethyl-17-alpha-ethinyl-17-hydroxygon-4,9,11-trien-3-one
- 13-Ethyl-17-hydroxy-18,19-dinor-17alpha-pregna-4,9,11-trien-20-yn-3-one
- 13-Ethyl-17α-ethynyl-17β-hydroxygona-4,9,11-trien-3-one
- 13-beta-Ethyl-17-alpha-ethinyl-17-hydroxy-gona-4,9,11-triene-3-one
- 18,19-Dinor-17-alpha-pregna-4,9,11-trien-20-yn-3-one, 13-ethyl-17-hydroxy-
- 18,19-Dinor-17α-pregna-4,9,11-trien-20-yn-3-one, 13-ethyl-17-hydroxy-
- 18,19-Dinorpregna-4,9,11-trien-20-yn-3-one, 13-ethyl-17-hydroxy-, (17-alpha)- (9CI)
- 18,19-Dinorpregna-4,9,11-trien-20-yn-3-one, 13-ethyl-17-hydroxy-, (17α)-
- See more synonyms
- A 46745
- Brn 5610726
- Dimetriose
- Dimetrose
- Ethylnorgestrienone
- Gestrigone
- Gestrinona
- Gestrinona [INN-Spanish]
- Gestrinone [USAN:INN:BAN]
- Gestrinonum
- Gestrinonum [INN-Latin]
- Nemestran
- Pregna-4,9,11-trien-20-yn-3-one, 13-ethyl-17-hydroxy-18,19-dinor-, (17alpha)-
- R-2323
- Ru 2323
- Tridomose
- Unii-1421533Rcm
- Gestrinone
