CAS 1643489-24-0

Tavapadon

Description:

Tavapadon is a novel chemical compound that acts as a selective dopamine D1 receptor agonist. It is primarily investigated for its potential therapeutic applications in treating conditions such as Parkinson's disease and other movement disorders. The compound is characterized by its ability to enhance dopaminergic signaling, which can help alleviate symptoms associated with dopamine deficiency. Tavapadon exhibits a favorable pharmacokinetic profile, including good oral bioavailability and a manageable half-life, making it suitable for clinical use. Its selectivity for the D1 receptor over other dopamine receptor subtypes is significant, as it may reduce the risk of side effects commonly associated with broader dopamine agonists. Additionally, ongoing research is focused on understanding its safety profile, efficacy, and optimal dosing regimens. As with many investigational drugs, further studies are essential to fully elucidate its mechanisms of action and therapeutic potential.

Formula: C₁₉H₁₆F₃N₃O₃

Synonyms:

• Tavapadon
• PF 6649751

(-)-1,5-Dimethyl-6-(2-methyl-4-((3-(trifluoromethyl)pyridin-2-yl)oxy)phenyl)pyrimidine-2,4(1H,3H)-dione

CAS: 1643489-24-0

Formula: C₁₉H₁₆F₃N₃O₃

Purity: 97%

Color and Shape: Solid

Molecular weight: 391.3438

Ref: IN-DA01LICI

(-)-1,5-Dimethyl-6-(2-Methyl-4-((3-(Trifluoromethyl)Pyridin-2-Yl)Oxy)Phenyl)Pyrimidine-2,4(1H,3H)-Dione

CAS: 1643489-24-0

(-)-1,5-Dimethyl-6-(2-Methyl-4-((3-(Trifluoromethyl)Pyridin-2-Yl)Oxy)Phenyl)Pyrimidine-2,4(1H,3H)-Dione

Purity: 97%

Molecular weight: 391.34g/mol

Ref: 54-PC108683

Tavapadon

CAS: 1643489-24-0

Tavapadon

Purity: ≥98%

Molecular weight: 391.34g/mol

Ref: 54-BUP09419

Tavapadon

CAS: 1643489-24-0

Tavapadon (CVL-751) is an orally active and highly selective dopamine D1/D5 receptor partial agonist.

Formula: C₁₉H₁₆F₃N₃O₃

Purity: 99.33% - 99.8%

Color and Shape: Solid

Molecular weight: 391.34

Ref: TM-T16999

Tavapadon

CAS: 1643489-24-0

Tavapadon is a peptide that binds to the GABAA receptor and enhances its activity. It is used as a research tool in cell biology and pharmacology, e.g., to study the effects of GABA on ion channels, ligand-receptor interactions, and antibody-antigen reactions. Tavapadon is also used as an inhibitor for certain types of protein interactions that are important for cell function.

Formula: C₁₉H₁₆F₃N₃O₃

Purity: Min. 95%

Molecular weight: 391.3 g/mol

Ref: 3D-TQC48924