CAS 1649-18-9
:Azaperone
Description:
Azaperone is a chemical compound classified as a butyrophenone derivative, primarily known for its use as a tranquilizer in veterinary medicine, particularly for swine. It exhibits antipsychotic and sedative properties, functioning as a dopamine antagonist. Azaperone is typically administered to reduce stress and aggression in animals, facilitating handling and transport. The compound is characterized by its relatively low solubility in water, which influences its formulation for administration. Its pharmacological effects are attributed to its ability to block dopamine receptors, particularly in the central nervous system, leading to sedation without significant respiratory depression. Azaperone is also noted for its relatively long duration of action, making it suitable for various veterinary applications. Safety and efficacy profiles have been established through studies, although its use is regulated and should be conducted under veterinary supervision to ensure appropriate dosing and minimize potential side effects. Overall, Azaperone plays a significant role in animal husbandry, contributing to the welfare of livestock during stressful situations.
Formula:C19H22FN3O
InChI:InChI=1S/C19H22FN3O/c20-17-8-6-16(7-9-17)18(24)4-3-11-22-12-14-23(15-13-22)19-5-1-2-10-21-19/h1-2,5-10H,3-4,11-15H2
InChI key:InChIKey=XTKDAFGWCDAMPY-UHFFFAOYSA-N
SMILES:C(CCC(=O)C1=CC=C(F)C=C1)N2CCN(CC2)C3=CC=CC=N3
Synonyms:- 1-(4-Fluorophenyl)-4-[4-(2-pyridinyl)-1-piperazinyl]-1-butanone
- 1-(4-Fluorophenyl)-4-[4-(Pyridin-2-Yl)Piperazin-1-Yl]Butan-1-One
- 1-Butanone, 1-(4-fluorophenyl)-4-[4-(2-pyridinyl)-1-piperazinyl]-
- 4-Fluoro-4-(4-(2-Pyridyl)Piperazin-1-Yl)Butyrophenone
- 4′-Fluoro-4-[4-(2-pyridyl)-1-piperazinyl]butyrophenone
- Butyrophenone, 4′-fluoro-4-[4-(2-pyridyl)-1-piperazinyl]-
- Fluoperidol
- NSC 170976
- R-1929
- Stresnil
- Suicalm
- See more synonyms
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Found 16 products.
AZAPERONE CRS
CAS:<p>AZAPERONE CRS</p>Formula:C19H22FN3OColor and Shape:White. Powder.Molecular weight:327.3959Azaperone
CAS:AzaperoneFormula:C19H22FN3OPurity:100.0%Color and Shape:Off-White. To. BeigeMolecular weight:327.17469Azaperone
CAS:Drugs containing a pyrimidine ring (whether or not hydrogenated) or piperazine ring in the structureFormula:C19H22FN3OColor and Shape:White PowderMolecular weight:327.174691-Butanone, 1-(4-fluorophenyl)-4-[4-(2-pyridinyl)-1-piperazinyl]-
CAS:Formula:C19H22FN3OPurity:98%Color and Shape:SolidMolecular weight:327.3959Azaperone
CAS:Formula:C19H22FN3OPurity:≥ 98.0%Color and Shape:White to light yellow or pale beige powderMolecular weight:327.40Azaperone 1000 µg/mL in Acetonitrile
CAS:Controlled ProductFormula:C19H22FN3OColor and Shape:ColourlessMolecular weight:327.40Azaperone
CAS:<p>Azaperone, a sedative and antiemetic veterinary tranquilizer, belongs to pyridinylpiperazine and butyrophenone classes.</p>Formula:C19H22FN3OPurity:98.73%Color and Shape:White Or Off-White CrystallineMolecular weight:327.41-(4-Fluorophenyl)-4-(4-(pyridin-2-yl)piperazin-1-yl)butan-1-one
CAS:Purity:95.0%Color and Shape:SolidMolecular weight:327.40301513671875Azaperone
CAS:Controlled Product<p>Applications Sedative; tranquilizer.<br> Not a dangerous good if item is equal to or less than 1g/ml and there is less than 100g/ml in the package<br>References Heykants, et al.: Arzneim.-Forsch., 21, 982 (1971), Stresser, D., et al.: Drug Metab. Dispos., 28, 1440 (2000), Egnell, A., et al.: J. Pharmacol. Exp. Ther., 305, 1251 (2003), Wester, M., et al.: J. Biol. Chem., 279, 35630 (2004),<br></p>Formula:C19H22FN3OColor and Shape:Off-White To BeigeMolecular weight:327.40Azaperone
CAS:<p>Azaperone is a potent sedative-hypnotic drug that is used to treat insomnia and as an aid in the treatment of acute, severe pain. It is also used to control convulsions in animals. Azaperone belongs to the class of barbiturates and has inhibitory effects on adrenal cortical activity and is therefore able to reduce the secretion of cortisol. In humans, it reduces the production of cortisol by inhibiting its release from the adrenal glands. Azaperone also stimulates ovulation in female mammals. The detection sensitivity for azaperone can be increased by using a LC-MS/MS method, which enables the measurement of picograms per millilitre (pg/mL) levels in human serum. This method was validated using monoclonal antibody (mAb) targeting azaperone and pentobarbital sodium, a structural heart disease marker with high analytical specificity for barbiturates.</p>Formula:C19H22FN3OPurity:Min. 95%Color and Shape:White PowderMolecular weight:327.4 g/molAzaperone (1 mg/mL in Methanol)
CAS:Controlled ProductFormula:C19H22FN3OColor and Shape:ColourlessMolecular weight:327.40Azaperone 100 µg/mL in Acetonitrile
CAS:Formula:C19H22FN3OColor and Shape:Single SolutionMolecular weight:327.40
![1-Butanone, 1-(4-fluorophenyl)-4-[4-(2-pyridinyl)-1-piperazinyl]-](/_next/image/?url=https%3A%2Fstatic.cymitquimica.com%2Fproducts%2FIN%2Fthumb%2FDA001V4Y.jpg&w=3840&q=75)
