CAS 170105-16-5

Imidafenacin

Description:

Imidafenacin is a chemical compound primarily used as a medication for the treatment of overactive bladder symptoms. It belongs to the class of drugs known as antimuscarinics, which work by inhibiting the action of acetylcholine on muscarinic receptors in the bladder, thereby reducing involuntary contractions and increasing bladder capacity. The molecular structure of Imidafenacin features a unique arrangement that contributes to its pharmacological activity, including a piperidine ring and various functional groups that enhance its selectivity and potency. It is typically administered orally and is characterized by its relatively long half-life, allowing for once-daily dosing in clinical settings. Common side effects may include dry mouth, constipation, and blurred vision, which are typical of antimuscarinic agents. Imidafenacin is notable for its balance between efficacy and tolerability, making it a valuable option in the management of urinary incontinence. As with any medication, it is essential to consider individual patient factors and potential drug interactions when prescribing Imidafenacin.

Formula: C₂₀H₂₁N₃O

InChI: InChI=1/C20H21N3O/c1-16-22-13-15-23(16)14-12-20(19(21)24,17-8-4-2-5-9-17)18-10-6-3-7-11-18/h2-11,13,15H,12,14H2,1H3,(H2,21,24)

InChI key: InChIKey=SQKXYSGRELMAAU-UHFFFAOYSA-N

SMILES: C(CCN1C(C)=NC=C1)(C(N)=O)(C2=CC=CC=C2)C3=CC=CC=C3

Synonyms:

• 1H-Imidazole-1-butanamide, 2-methyl-α,α-diphenyl-
• 2-Methyl-α,α-diphenyl-1H-imidazole-1-butanamide
• 4-(2-Methyl-1-imidazolyl)-2,2-diphenylbutanamide
• 4-(2-Methyl-1H-Imidazol-1-Yl)-2,2-Diphenylbutanamide
• Krp 197
• Ono 8025
• Staybla
• Uritos
• Imidafenacin
• Midana new API
• 4-(2-methylimidazol-1-yl)-2,2-diphenylbutanamide
• IMidafenacin DISCONTINUED-PATENTED PRODUCT
• KRP-197; ONO-8025
• )-2,2-diphenyL
• diphenylbutanaMide
• 4-(2-methyL
• Imidafenacin-d10

Imidafenacin

CAS: 170105-16-5

Formula: C₂₀H₂₁N₃O

Purity: 98%

Color and Shape: Solid

Molecular weight: 319.4002

Ref: IN-DA00ABKE

4-(2-Methyl-1H-Imidazol-1-Yl)-2,2-Diphenylbutanamide

CAS: 170105-16-5

4-(2-Methyl-1H-Imidazol-1-Yl)-2,2-Diphenylbutanamide

Purity: 98%

Molecular weight: 319.4g/mol

Ref: 54-OR1026599

Imidafenacin

CAS: 170105-16-5

Imidafenacin

Purity: ≥98%

Molecular weight: 319.4g/mol

Ref: 54-BUP11325

Imidafenacin

CAS: 170105-16-5

Formula: C₂₀H₂₁N₃O

Color and Shape: White To Off-White Solid

Molecular weight: 319.41

Ref: 4Z-I-461

Imidafenacin-d10

CAS: 170105-16-5

Formula: C₂₀H₁₁D₁₀N₃O

Color and Shape: White To Off-White Solid

Molecular weight: 329.47

Ref: 4Z-I-4622

Imidafenacin

CAS: 170105-16-5

Imidafenacin (KRP-197)(KRP-197; ONO-8025) is a potent and selective inhibitor of M3 receptors with Kb of 0.317 nM.

Formula: C₂₀H₂₁N₃O

Purity: 99.17%

Color and Shape: Solid

Molecular weight: 319.4

Ref: TM-T4986

Imidafenacin

CAS: 170105-16-5

Antagonist of muscarinic (M3) receptor

Formula: C₂₀H₂₁N₃O

Purity: Min. 95%

Color and Shape: White to off-white solid.

Molecular weight: 319.16846

Ref: 3D-FI24546

Imidafenacin-d13

Controlled Product

CAS: 170105-16-5

Formula: C₂₀D₁₃H₈N₃O

Color and Shape: Neat

Molecular weight: 332.48

Ref: TR-I275014

Imidafenacin-d10

Controlled Product

CAS: 170105-16-5

Formula: C₂₀D₁₀H₁₁N₃O

Color and Shape: Neat

Molecular weight: 329.462

Ref: TR-I275013