CAS 176324-85-9

2-[(4-Bromophenyl)methyl]-4,5-dihydro-4,4-dimethyloxazole

Controlled Product

CAS: 176324-85-9

Applications 2-[(4-Bromophenyl)methyl]-4,5-dihydro-4,4-dimethyloxazole is an intermediate used in the synthesis of Bilastine-d6 (B385002), which is labelled Bilastine. It is a novel, nonsedating H1-antihistamine developed for symptomatic treatment of allergic rhinitis and chronic idiopathic urticaria.
References Van Cauwenberge, P., et al.: Clin. Exp. Allergy, 30, 891 (2000), Bauchau, V., et al.: Eur. Respir. J., 24, 758 (2004), Lehman, J., et al.: Drugs, 66, 2309 (2006),

Formula: C₁₂H₁₄BrNO

Color and Shape: Neat

Molecular weight: 268.15

Ref: TR-B711005