CAS 177834-92-3

Eletriptan hydrobromide

Description:

Eletriptan hydrobromide is a pharmaceutical compound primarily used as a medication for the acute treatment of migraine headaches. It belongs to the class of drugs known as triptans, which are selective agonists for serotonin receptors, specifically the 5-HT_1B and 5-HT_1D subtypes. This action helps to alleviate migraine symptoms by causing vasoconstriction of cranial blood vessels and inhibiting the release of pro-inflammatory neuropeptides. The substance is typically administered in oral form and is characterized by its relatively rapid onset of action. In terms of its chemical properties, eletriptan hydrobromide is a white to off-white crystalline powder, soluble in water, and has a specific molecular structure that contributes to its pharmacological effects. It is important to note that, like other medications, eletriptan hydrobromide may have side effects, including dizziness, fatigue, and sensations of tingling or warmth. As with any medication, it should be used under the guidance of a healthcare professional.

Formula: C₂₂H₂₆N₂O₂S

InChI: InChI=1/C22H26N2O2S.BrH/c1-24-12-5-6-19(24)15-18-16-23-22-10-9-17(14-21(18)22)11-13-27(25,26)20-7-3-2-4-8-20;/h2-4,7-10,14,16,19,23H,5-6,11-13,15H2,1H3;1H/t19-;/m1./s1

InChI key: InChIKey=UTINOWOSWSPFLJ-FSRHSHDFSA-N

SMILES: C(C=1C=2C(NC1)=CC=C(CCS(=O)(=O)C3=CC=CC=C3)C2)[C@@H]4N(C)CCC4.Br

Synonyms:

• (R)-5-[2-(Benzenesulfonyl)ethyl]-3-[(N-methylpyrrolidin-2-yl)methyl]-1H-indole hydrobromide
• 1H-Indole, 3-[(1-methyl-2-pyrrolidinyl)methyl]-5-[2-(phenylsulfonyl)ethyl]-, monohydrobromide, (R)-
• 1H-Indole, 3-[[(2R)-1-methyl-2-pyrrolidinyl]methyl]-5-[2-(phenylsulfonyl)ethyl]-, hydrobromide (1:1)
• 1H-Indole, 3-[[(2R)-1-methyl-2-pyrrolidinyl]methyl]-5-[2-(phenylsulfonyl)ethyl]-, monohydrobromide
• 3-(((2R)-1-Methyl-2-Pyrrolidinyl))Methyl)-5-(2-(Phenylsulfonyl)Ethyl)-1H-Indole Hydrobromide
• 3-[(1-methylpyrrolidin-2-yl)methyl]-5-[2-(phenylsulfonyl)ethyl]-1H-indole hydrobromide (1:1)
• 3-{[(2R)-1-methylpyrrolidin-2-yl]methyl}-5-[2-(phenylsulfonyl)ethyl]-1H-indole hydrobromide (1:1)
• Eletriptan Base
• Eletriptan Hbr
• Relert
• Relpax
• Uk 116044-04
• Eletriptan hydrobromide
• Eletriptan-d3 HBr
• QR-2008082103-ELCPT
• Also see: E505000
• Eletriptan HCl
• Eletriptan hydrobromide (Eletriptan HBr)
• (R)-3-((1-Methylpyrrolidin-2-yl)Methyl)-5-(2-(phenylsulfonyl)ethyl)-1H-indole hydrobroMide
• Eletriptan hydrobromide USP/EP/BP
• Unii-m41W832ta3
• etriptan hydrobromide
• Eletriptan hydrobromide, 99%, a selective 5-HT1B/1D receptor agonist
• 5-[2-(benzenesulfonyl)ethyl]-3-[[(2R)-1-methyl-2-pyrrolidinyl]methyl]-1H-indole hydrobromide

1H-Indole, 3-[[(2R)-1-methyl-2-pyrrolidinyl]methyl]-5-[2-(phenylsulfonyl)ethyl]-, hydrobromide (1:1)

CAS: 177834-92-3

Formula: C₂₂H₂₇BrN₂O₂S

Purity: 98%

Color and Shape: Solid

Molecular weight: 463.4310

Ref: IN-DA0025L1

Eletriptan hydrobromide

CAS: 177834-92-3

Eletriptan hydrobromide (Eletriptan HBr) is an orally active agonist with specific affinity for the 5-hydroxytriptamine1B/1D receptor.

Formula: C₂₂H₂₇BrN₂O₂S

Purity: 99.69% - 99.85%

Color and Shape: Tan Solid

Molecular weight: 463.43

Ref: TM-T0216

Eletriptan hydrobromide

CAS: 177834-92-3

Eletriptan hydrobromide

Purity: ≥95%

Molecular weight: 463.43g/mol

Ref: 54-BUP15007

Eletriptan hydrobromide

CAS: 177834-92-3

Formula: C₂₂H₂₆N₂O₂S·HBr

Purity: ≥ 97.0%

Color and Shape: White to off-white powder

Molecular weight: 463.43

Ref: 7W-GK9539

(R)-3-((1-Methylpyrrolidin-2-Yl)Methyl)-5-(2-(Phenylsulfonyl)Ethyl)-1H-Indole Hydrobromide

CAS: 177834-92-3

(R)-3-((1-Methylpyrrolidin-2-Yl)Methyl)-5-(2-(Phenylsulfonyl)Ethyl)-1H-Indole Hydrobromide

Purity: 98%

Molecular weight: 463.43g/mol

Ref: 54-OR1029414

Eletriptan HBr

CAS: 177834-92-3

Formula: C₂₂H₂₆N₂O₂S·HBr

Color and Shape: Pale Yellow Solid

Molecular weight: 382.52 80.91

Ref: 4Z-E-121

Eletriptan Hydrobromide

Controlled Product

CAS: 177834-92-3

Formula: C₂₂H₂₆N₂O₂S·BrH

Color and Shape: Neat

Molecular weight: 463.43

Ref: 86-MM3542.00

Relpax

Controlled Product

CAS: 177834-92-3

Applications Relpax is a second generation triptan drug used in the treatment of migraine headaches.
References McCormack, P.L. et al.: Drugs, 66, 1129 (2006); Goadsby, P.J. et al.: Neurology, 54, 156 (2000); Napier, C. et al.: Eur. J. Pharmacol., 368, 259 (1999);

Formula: C₂₂H₂₆N₂O₂S·BrH

Color and Shape: Neat

Molecular weight: 463.43

Ref: TR-R143400

Eletriptan HBr - Bio-X ™

CAS: 177834-92-3

Eletriptan is a triptan drug used for the treatment of migraines. This drug is an agonist of serotonin receptors, mainly 5-HT 1B/D. It acts to relieve migraines by causing vasoconstriction in intracranial blood vessels.

Formula: C₂₂H₂₇N₂O₂SBr

Purity: Min. 95%

Color and Shape: Powder

Molecular weight: 481.45 g/mol

Ref: 3D-FE162187

Eletriptan hydrobromide

CAS: 177834-92-3

Agonist of 5-HT1B/D serotonin receptors; anti-migraine medication

Formula: C₂₂H₂₆N₂O₂S•HBr

Purity: Min. 95%

Color and Shape: Powder

Molecular weight: 481.45 g/mol

Ref: 3D-FE38878