CAS 179756-85-5

Eptapirone

Description:

Eptapirone is a chemical compound classified as a selective serotonin receptor agonist, specifically targeting the 5-HT1A receptor. It is primarily investigated for its potential therapeutic applications in treating anxiety and depression. Eptapirone is known for its anxiolytic properties, which may arise from its ability to enhance serotonin neurotransmission in the brain. The compound has a relatively complex molecular structure, which contributes to its pharmacological activity. In terms of solubility, eptapirone is typically soluble in organic solvents, but its solubility in water may be limited. The compound has undergone various preclinical and clinical studies to evaluate its efficacy and safety profile. As with many psychoactive substances, the pharmacokinetics of eptapirone, including its absorption, distribution, metabolism, and excretion, are crucial for understanding its therapeutic potential and side effects. Overall, eptapirone represents a promising avenue in the development of novel treatments for mood disorders, although further research is necessary to fully elucidate its mechanisms of action and clinical utility.

Formula: C₁₆H₂₃N₇O₂·C₄H₄O₄

InChI: InChI=1S/C16H23N7O2.C4H4O4/c1-20-14(24)13-19-23(16(20)25)8-3-2-7-21-9-11-22(12-10-21)15-17-5-4-6-18-15;5-3(6)1-2-4(7)8/h4-6,13H,2-3,7-12H2,1H3;1-2H,(H,5,6)(H,7,8)/b;2-1+

InChI key: InChIKey=IRTCWPNSLGQHOR-WLHGVMLRSA-N

SMILES: C(CCCN1C(=O)N(C)C(=O)C=N1)N2CCN(CC2)C=3N=CC=CN3.C(=C/C(O)=O)\C(O)=O

Synonyms:

• 1,2,4-Triazine-3,5(2H,4H)-dione, 4-methyl-2-[4-[4-(2-pyrimidinyl)-1-piperazinyl]butyl]-, (2E)-2-butenedioate (1:1)
• Eptapirone
• 1,2,4-Triazine-3,5(2H,4H)-dione, 4-methyl-2-[4-[4-(2-pyrimidinyl)-1-piperazinyl]butyl]-, (E)-2-butenedioate (1:1)

Eptapirone

CAS: 179756-85-5

Eptapirone is a peptide that binds to the β-adrenergic receptor, which is a G protein-coupled receptor. This receptor has been found in many tissues in the body, including the heart and brain. Eptapirone can be used as a research tool for studying the function of these receptors in these tissues. It also has been shown to have an inhibitory effect on ion channels and can be used as an antibody ligand.

Formula: C₁₆H₂₃N₇O₂

Purity: Min. 95%

Molecular weight: 345.4 g/mol

Ref: 3D-EHA75685

Eptapirone fumarate

CAS: 179756-85-5

Eptapirone (F11440) is a strong 5HT1A agonist with high anxiolytic and antidepressant effects, more potent than buspirone and flesinoxan.

Formula: C₂₀H₂₇N₇O₆

Color and Shape: Solid

Molecular weight: 461.479

Ref: TM-T70183