CAS 185913-78-4

Satavaptan

Description:

Satavaptan is a chemical compound classified as a selective vasopressin V2 receptor antagonist, primarily used in the treatment of conditions associated with water retention, such as hyponatremia and heart failure. Its molecular structure features a unique arrangement of atoms that contributes to its pharmacological properties. Satavaptan is known for its ability to inhibit the action of vasopressin, a hormone that regulates water balance in the body, thereby promoting diuresis and reducing fluid overload. The compound is typically administered in oral form and has been studied for its potential benefits in managing various disorders related to fluid retention. In terms of solubility, Satavaptan exhibits moderate solubility in organic solvents, which is relevant for its formulation in pharmaceutical preparations. Safety and efficacy profiles are evaluated through clinical trials, and like many medications, it may have side effects that require monitoring. Overall, Satavaptan represents a significant advancement in the therapeutic management of conditions linked to abnormal water retention.

Formula: C₃₃H₄₅N₃O₈S

InChI: InChI=1/C33H45N3O8S/c1-6-43-25-8-9-27-26(22-25)33(13-11-24(12-14-33)44-20-17-35-15-18-42-19-16-35)31(38)36(27)45(39,40)29-10-7-23(21-28(29)41-5)30(37)34-32(2,3)4/h7-10,21-22,24H,6,11-20H2,1-5H3,(H,34,37)/t24-,33+

InChI key: InChIKey=QKXJWFOKVQWEDZ-VCCCEUOBNA-N

SMILES: O=C1[C@]2(C=3C(N1S(=O)(=O)C4=C(OC)C=C(C(NC(C)(C)C)=O)C=C4)=CC=C(OCC)C3)CC[C@H](OCCN5CCOCC5)CC2

Synonyms:

• Benzamide, N-(1,1-dimethylethyl)-4-[[5′-ethoxy-4-[2-(4-morpholinyl)ethoxy]-2′-oxospiro[cyclohexane-1,3′-[3H]indol]-1′(2′H)-yl]sulfonyl]-3-methoxy-, cis-
• SR 121463
• Benzamide, N-(1,1-dimethylethyl)-4-[[cis-5′-ethoxy-4-[2-(4-morpholinyl)ethoxy]-2′-oxospiro[cyclohexane-1,3′-[3H]indol]-1′(2′H)-yl]sulfonyl]-3-methoxy-
• Satavaptan
• N-(1,1-Dimethylethyl)-4-[[cis-5′-ethoxy-4-[2-(4-morpholinyl)ethoxy]-2′-oxospiro[cyclohexane-1,3′-[3H]indol]-1′(2′H)-yl]sulfonyl]-3-methoxybenzamide

Ibrexafungerp

CAS: 185913-78-4

Ibrexafungerp

Purity: ≥98%

Molecular weight: 730.03g/mol

Ref: 54-BUP20662

Satavaptan

CAS: 185913-78-4

Satavaptan is a vasopressin V2 receptor antagonist. Satavaptan improves the control of ascites in cirrhosis.

Formula: C₃₃H₄₅N₃O₈S

Color and Shape: Solid

Molecular weight: 643.79

Ref: TM-T28664