CAS 190786-44-8: Bepotastine besilate
Description:Bepotastine besilate is an antihistamine medication primarily used for the treatment of allergic conjunctivitis and other allergic conditions. It functions as a selective H1 receptor antagonist, effectively blocking the action of histamine, a compound involved in allergic responses. This substance is characterized by its ability to alleviate symptoms such as itching, redness, and swelling associated with allergies. Bepotastine besilate is typically administered as an ophthalmic solution, allowing for direct application to the eyes, which enhances its efficacy and minimizes systemic side effects. The compound is known for its rapid onset of action and relatively favorable safety profile, making it a preferred choice in allergy management. Additionally, it is soluble in water, which facilitates its formulation in liquid dosage forms. As with any medication, potential side effects may include local irritation or discomfort, but these are generally mild. Overall, bepotastine besilate represents a targeted approach to managing allergic symptoms, particularly in the ocular region.
Formula:C21H25ClN2O3·C6H6O3S
InChI:InChI=1S/C21H25ClN2O3.C6H6O3S/c22-17-8-6-16(7-9-17)21(19-4-1-2-12-23-19)27-18-10-14-24(15-11-18)13-3-5-20(25)26;7-10(8,9)6-4-2-1-3-5-6/h1-2,4,6-9,12,18,21H,3,5,10-11,13-15H2,(H,25,26);1-5H,(H,7,8,9)/t21-;/m0./s1
InChI key:InChIKey=UDGHXQPQKQPSBB-BOXHHOBZSA-N
SMILES:O=C(O)CCCN1CCC(OC(C2=NC=CC=C2)C3=CC=C(Cl)C=C3)CC1.O=S(=O)(O)C=1C=CC=CC1
- Synonyms:
- 1-Piperidinebutanoic acid, 4-[(4-chlorophenyl)-2-pyridinylmethoxy]-, (S)-, monobenzenesulfonate
- Talion
- 1-Piperidinebutanoic acid, 4-[(S)-(4-chlorophenyl)-2-pyridinylmethoxy]-, benzenesulfonate (1:1)
- Bepotastine besilate
- 1-Piperidinebutanoic acid, 4-[(S)-(4-chlorophenyl)-2-pyridinylmethoxy]-, monobenzenesulfonate