CAS 192374-14-4

Radafaxine

Description:

Radafaxine, identified by its CAS number 192374-14-4, is a chemical compound that belongs to the class of phenethylamines. It is primarily recognized for its potential use as a stimulant and has been investigated for its effects on the central nervous system. The substance is characterized by its ability to enhance neurotransmitter activity, particularly dopamine and norepinephrine, which may contribute to its stimulant properties. Radafaxine has been studied for its potential applications in treating conditions such as attention deficit hyperactivity disorder (ADHD) and narcolepsy. Its pharmacological profile suggests a mechanism of action that may involve the inhibition of reuptake of certain neurotransmitters, leading to increased levels in the synaptic cleft. However, as with many compounds in this class, the safety, efficacy, and long-term effects of Radafaxine require thorough investigation through clinical trials. As of the latest data, it remains a subject of research rather than a widely approved therapeutic agent.

Formula: C₁₃H₁₈ClNO₂

InChI: InChI=1S/C13H18ClNO2/c1-9-13(16,17-8-12(2,3)15-9)10-5-4-6-11(14)7-10/h4-7,9,15-16H,8H2,1-3H3/t9-,13+/m0/s1

InChI key: InChIKey=RCOBKSKAZMVBHT-TVQRCGJNSA-N

SMILES: O[C@@]1([C@H](C)NC(C)(C)CO1)C2=CC(Cl)=CC=C2

Synonyms:

• 2-Morpholinol, 2-(3-chlorophenyl)-3,5,5-trimethyl-, (2S,3S)-
• (+)-(2S,3S)-2-(3-chlorophenyl)-3,5,5-trimethyl-2-morpholinol
• (2S,3S)-2-(3-Chlorophenyl)-3,5,5-trimethyl-2-morpholinol
• 2-Morpholinol, 2-(3-chlorophenyl)-3,5,5-trimethyl-, (2S-cis)-
• Radafaxine

2-Morpholinol, 2-(3-chlorophenyl)-3,5,5-trimethyl-, (2S,3S)-

CAS: 192374-14-4

Formula: C₁₃H₁₉Cl₂NO₂

Color and Shape: Solid

Molecular weight: 292.2015

Ref: IN-DA002FV4

(S,S)-Hydroxy Bupropion

CAS: 192374-14-4

Formula: C₁₃H₁₈ClNO₂

Color and Shape: White To Off-White Solid

Molecular weight: 255.74

Ref: 4Z-B-0523

(S,S)-Hydroxy Bupropion

CAS: 192374-14-4

Applications (S,S) Enantiomer metabolite of Bupropion (B689625), an antidepressant.
References Hsyu, P-H., et al.: J. Clin. Pharm., 37, 737 (1997), Rotzinger, S., et al.: Cellular & Mol. Neurobiology, 19, 4, 427 (1999); US 6342496

Formula: C₁₃H₁₈ClNO₂·ClH

Color and Shape: Neat

Molecular weight: 292.20

Ref: TR-H830670

(S,S)-Hydroxy bupropion

CAS: 192374-14-4

(S,S)-Hydroxy bupropion is a drug that is used to treat some forms of depression in humans. It is a dopaminergic agent that acts on the dopamine receptor and has been shown to be effective for the treatment of some metabolic disorders in humans. The low potency of this drug may be due to its metabolism by CYP2B6, which prevents it from being active when taken orally. This drug also has been shown to have antagonist effects against the cannabinoid receptor (CB1) and may have therapeutic potential for treating obesity and nicotine addiction.

Formula: C₁₃H₁₈ClNO₂

Purity: Min. 95%

Molecular weight: 255.74 g/mol

Ref: 3D-FH23926

(S,S)-Hydroxy Bupropion

CAS: 192374-14-4

Formula: C₁₃H₁₈ClNO₂

Molecular weight: 255.74

Ref: ST-EA-CP-B21029