CAS 2010159-47-2

MZP-54

Description:

MZP-54, identified by its CAS number 2010159-47-2, is a synthetic compound that belongs to a class of substances known for their potential psychoactive effects. While specific characteristics such as its molecular formula, structure, and physical properties may not be widely documented, compounds in this category often exhibit properties that can influence neurotransmitter systems in the brain. MZP-54 may interact with serotonin receptors, similar to other substances in its class, which can lead to various psychological effects. As with many novel compounds, research on MZP-54 is limited, and its safety profile, pharmacokinetics, and long-term effects are not well established. It is crucial to approach such substances with caution, as their legal status and potential for abuse can vary significantly across different jurisdictions. Always refer to reliable sources and scientific literature for the most accurate and up-to-date information regarding any chemical substance.

Formula: C₅₅H₆₆ClN₇O₉S

InChI: InChI=1S/C55H66ClN7O9S/c1-34-27-46(60-43-18-16-42(56)17-19-43)45-28-41(15-20-47(45)63(34)36(3)64)38-11-13-40(14-12-38)52(67)57-21-22-70-23-24-71-25-26-72-32-49(66)61-51(55(4,5)6)54(69)62-31-44(65)29-48(62)53(68)58-30-37-7-9-39(10-8-37)50-35(2)59-33-73-50/h7-20,28,33-34,44,46,48,51,60,65H,21-27,29-32H2,1-6H3,(H,57,67)(H,58,68)(H,61,66)/t34-,44+,46+,48-,51+/m0/s1

InChI key: InChIKey=FYSWLIFIYIVHPI-DDWISSAJSA-N

SMILES: N([C@H]1C=2C(N(C(C)=O)[C@@H](C)C1)=CC=C(C2)C3=CC=C(C(NCCOCCOCCOCC(N[C@H](C(=O)N4[C@H](C(NCC5=CC=C(C=C5)C=6SC=NC6C)=O)C[C@@H](O)C4)C(C)(C)C)=O)=O)C=C3)C7=CC=C(Cl)C=C7

Synonyms:

• MZP-54

(2S,4R)-1-[(2S)-2-[2-(2-{2-[2-({4-[(2S,4R)-1-acetyl-4-[(4-chlorophenyl)amino]-2-methyl-1,2,3,4-tetrahydroquinolin-6-yl]phenyl}formamido)ethoxy]ethoxy}ethoxy)acetamido]-3,3-dimethylbutanoyl]-4-hydroxy-N-{[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl}pyrrolidine-2-carboxamide

CAS: 2010159-47-2

Formula: C₅₅H₆₆ClN₇O₉S

Purity: 98.16%

Molecular weight: 1036.6720

Ref: IN-DA01ENX4

MZP-54

CAS: 2010159-47-2

MZP-54 is a selective degrader of BRD3/4 based on PROTAC technology(Kd of 4 nM for Brd4BD2)

Formula: C₅₅H₆₆ClN₇O₉S

Purity: 98%

Color and Shape: Solid

Molecular weight: 1036.67

Ref: TM-T13785

MZP-54

CAS: 2010159-47-2

MZP-54 is a natural product that inhibits the HIV virus. It binds to HIV-1 integrase and blocks the integration of viral DNA into the host cell genome. MZP-54 has been shown to inhibit tumor growth in vitro and in vivo, as well as to reduce the number of cancer cells in culture. It also inhibits angiogenesis and has shown activity against a variety of human cancers, including prostate, breast, colon, lung, leukemia, and lymphoma. MZP-54 also inhibits expression of genes regulated by bromodomain proteins. Bromodomain proteins are involved in regulating gene expression by binding to acetylated lysine residues on histones H3 and H4. This protein is expressed at high levels in heart tissue and is associated with cardiotoxicity caused by coronary heart disease or heart failure. In addition, MZP-54 has been found to inhibit renal fibrosis and regulate erythropoietin production.

Formula: C₅₅H₆₆ClN₇O₉S

Purity: Min. 95%

Molecular weight: 1,036.67 g/mol

Ref: 3D-KFD15947