CAS 2056122-11-1

Thieno[2,3-b]pyridin-6(7H)-one, 4-amino-5-[6-(4-methyl-1-piperazinyl)-1H-benzimidazol-2-yl]-

Description:

Thieno[2,3-b]pyridin-6(7H)-one, 4-amino-5-[6-(4-methyl-1-piperazinyl)-1H-benzimidazol-2-yl]- is a complex organic compound characterized by its unique bicyclic structure that incorporates both thieno and pyridine moieties. The presence of an amino group and a benzimidazole derivative contributes to its potential biological activity, making it of interest in medicinal chemistry. The compound features a piperazine ring, which is often associated with pharmacological properties, enhancing its interaction with biological targets. Its molecular structure suggests potential applications in drug development, particularly in areas such as oncology or neurology, where compounds with such structural features may exhibit therapeutic effects. The compound's solubility, stability, and reactivity would depend on its specific functional groups and overall molecular conformation. As with many synthetic organic compounds, understanding its characteristics, including melting point, boiling point, and spectral properties, would be essential for further applications and studies.

Formula: C₁₉H₂₀N₆OS

Synonyms:

• Thieno[2,3-b]pyridin-6(7H)-one, 4-amino-5-[6-(4-methyl-1-piperazinyl)-1H-benzimidazol-2-yl]-
• 4-Amino-5-(6-(4-methylpiperazin-1-yl)-1H-benzo[d]imidazol-2-yl)thieno[2,3-b]pyridin-6(7H)-one
• HPK1-IN-2
• HPK1-IN-2 dihydrochloride
• Thieno[2,3-b]pyridin-6(7H)-one, 4-amino-5-[6-(4-methyl-1-piperazinyl)-1H-benzimidazol-2-yl]-HPK1-IN-2

HPK1-IN-2

CAS: 2056122-11-1

HPK1-IN-2

Purity: ≥95%

Molecular weight: 380.47g/mol

Ref: 54-BUP08260

HPK1-IN-2

CAS: 2056122-11-1

HPK1-IN-2 is a strong, oral HPK1 inhibitor (IC50<0.05 μM), also blocking Lck, Flt3 kinases, with anticancer properties.

Formula: C₁₉H₂₀N₆OS

Purity: 97.31%

Color and Shape: Solid

Molecular weight: 380.47

Ref: TM-T9017

HPK1-IN-2 dihydrochloride

CAS: 2056122-11-1

HPK1-IN-2 is a peptide that belongs to the group of activators. It is a potent inhibitor of potassium channels and has been shown to activate calcium channels. HPK1-IN-2 is also an antibody that can be used in research tools for cell biology and pharmacology. This peptide can be used to study protein interactions, such as those between ion channels and receptors, ligands, or proteins. HPK1-IN-2 has been shown to inhibit potassium channels, which are involved in the regulation of cellular excitability and neurotransmitter release.

Formula: C₁₉H₂₀N₆OS

Purity: Min. 95%

Molecular weight: 380.5 g/mol

Ref: 3D-GHD12211