CAS 2158266-58-9

GNE-207

CAS: 2158266-58-9

GNE-207 is a peptide that selectively binds to the extracellular domain of the human erythropoietin receptor (EPOR) and is a potent EPOR activator. GNE-207 has been shown to inhibit tumor growth in xenograft models, as well as to reduce vascular permeability in animal models. In vitro, GNE-207 inhibits proliferation of human tumor cells and induces apoptosis. GNE-207 is also an inhibitor of angiogenesis, which may be related to its ability to inhibit endothelial cell proliferation and migration.

Formula: C₂₉H₃₀N₆O₃

Purity: Min. 95%

Molecular weight: 510.6 g/mol

Ref: 3D-ILD26658

GNE-207

CAS: 2158266-58-9

GNE-207 is a selective and orally bioavailable inhibitor of the bromodomain of CBP (IC50: 1 nM).

Formula: C₂₉H₃₀N₆O₃

Purity: 98%

Color and Shape: Solid

Molecular weight: 510.59

Ref: TM-T15399