CAS 216853-59-7

NS3861

CAS: 216853-59-7

NS3861

Purity: ≥98%

Molecular weight: 284.22g/mol

Ref: 54-BUP10969

NS3861

CAS: 216853-59-7

NS3861 is a selective agonist for α3β4/α4β2 nAChRs, preferring β-subunits, with no effect on α4-based receptors.

Formula: C₁₂H₁₄BrNS

Purity: 99.853%

Color and Shape: Solid

Molecular weight: 284.22

Ref: TM-T9542

3-(3-Bromo-2-thienyl)-8-methyl-8-azabicyclo[3.2.1]oct-2-ene

CAS: 216853-59-7

3-(3-Bromo-2-thienyl)-8-methyl-8-azabicyclo[3.2.1]oct-2-ene is a competitive antagonist of the serotonin 5HT1A receptor and a selective competitive antagonist of the histamine H3 receptor. It has been shown to be an agonist at the alpha 2C adrenergic receptor and to have neuroprotective effects against glutamate toxicity in cultured hippocampal neurons. 3-(3-Bromo-2-thienyl)-8-methyl-8-azabicyclo[3.2.1]oct-2-ene is also a ligand for the LPA1 receptor, which may contribute to its antiinflammatory effects in vivo.

Formula: C₁₂H₁₄BrNS

Purity: Min. 95%

Molecular weight: 284.22 g/mol

Ref: 3D-RIA85359