CAS 224785-87-9

Piperazine,1-[[3-(1,4-dihydro-5-methyl-4-oxo-7-propylimidazo[5,1-f][1,2,4]triazin-2-yl)-4-ethoxyphenyl]sulfonyl]-4-methyl-

Description:

Piperazine, 1-[[3-(1,4-dihydro-5-methyl-4-oxo-7-propylimidazo[5,1-f][1,2,4]triazin-2-yl)-4-ethoxyphenyl]sulfonyl]-4-methyl- is a complex organic compound characterized by its piperazine core, which is a six-membered ring containing two nitrogen atoms. This compound features a sulfonyl group, which enhances its solubility and reactivity, and is substituted with a phenyl group that carries an ethoxy group and an imidazotriazine moiety. The presence of the imidazo[5,1-f][1,2,4]triazin structure suggests potential biological activity, possibly as an antimicrobial or anticancer agent, due to the known properties of similar compounds. The methyl and propyl groups contribute to the lipophilicity of the molecule, potentially influencing its pharmacokinetic properties. Overall, this compound's unique structure may offer interesting avenues for research in medicinal chemistry, particularly in the development of new therapeutic agents. However, specific biological activities and applications would require further investigation through experimental studies.

Formula: C₂₂H₃₀N₆O₄S

N-Desethyl-N-Methyl Vardenafil

CAS: 224785-87-9

Formula: C₂₂H₃₀N₆O₄S

Color and Shape: White To Off-White Solid

Molecular weight: 474.58

Ref: 4Z-V-0528

N-Desethyl-N-Methyl Vardenafil

CAS: 224785-87-9

Formula: C₂₂H₃₀N₆O₄S

Molecular weight: 474.58

Ref: ST-EA-CP-V28020

N-desethyl-N-methyl Vardenafil

CAS: 224785-87-9

N-Desethyl-N-methyl Vardenafil, a potential impurity in commercial vardenafil preparations, functions as a phosphodiesterase 5 (PDE5) inhibitor, similar to its parent compound. With an IC50 value of 2 nM, it exhibits potent inhibitory activity against PDE5.

Formula: C₂₂H₃₀N₆O₄S

Color and Shape: Solid

Molecular weight: 474.58

Ref: TM-T84929