CAS 2409964-40-3

2-Buten-1-amine, 3-fluoro-4-(phenylsulfonyl)-, hydrochloride (1:1), (2Z)-

Description:

2-Buten-1-amine, 3-fluoro-4-(phenylsulfonyl)-, hydrochloride (1:1), (2Z)- is a chemical compound characterized by its specific structural features and functional groups. It contains a butenamine backbone, which is an unsaturated amine, indicating the presence of both an amine (-NH2) and a double bond within its structure. The compound is further modified by the presence of a fluorine atom at the 3-position and a phenylsulfonyl group at the 4-position, which contributes to its reactivity and potential applications in medicinal chemistry. The hydrochloride salt form suggests enhanced solubility in water, making it suitable for various biological assays. The (2Z) designation indicates the specific geometric configuration of the double bond, which can influence the compound's biological activity and interaction with other molecules. Overall, this compound may exhibit unique properties due to its structural complexity, making it of interest in pharmaceutical research and development.

Formula: C₁₀H₁₂FNO₂S·ClH

Synonyms:

• 2-Buten-1-amine, 3-fluoro-4-(phenylsulfonyl)-, hydrochloride (1:1), (2Z)-

PXS-4787 hydrochloride

CAS: 2409964-40-3

PXS-4787 hydrochloride is a specific and potent pan-lysyl oxidase inhibitor that effectively eliminates the activity of lysyl oxidase. It exhibits varying IC50 values against different forms of the enzyme, including 2 μM (Bovine LOX), 3.2 μM (rh LOXL1), 0.6 μM (rh LOXL2), 1.4 μM (rh LOXL3), and 0.2 μM (rh LOXL4). In addition, PXS-4787 hydrochloride reduces the deposition and cross-linking of collagen I secreted by human fibroblasts.

Formula: C₁₀H₁₃ClFNO₂S

Color and Shape: Solid

Molecular weight: 265.73

Ref: TM-T201314