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CAS 2412715-30-9

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  • ERβ agonist-1

    CAS:
    <p>ERβagonist-1 (Compound 8) functions as a dual-active selective ERβ agonist (EC50: 46.8 nM) and an AR antagonist (IC50: 1555 nM). By binding to ERβ, it activates its signaling pathways while simultaneously inhibiting AR activity. Retaining selective ERβ agonist activity in mouse models, ERβagonist-1 is applicable in prostate cancer research.</p>
    Formula:C25H36O2
    Color and Shape:Solid
    Molecular weight:368.55