CymitQuimica logo

CAS 24359-22-6

:

Pizotifen maleate

Description:
Pizotifen maleate is a pharmaceutical compound primarily used as an antihistamine and a preventive treatment for migraines. It is classified as a serotonin receptor antagonist, specifically targeting the 5-HT2 receptor, which contributes to its efficacy in reducing migraine frequency. The maleate salt form enhances its solubility and stability, making it suitable for oral administration. Pizotifen is known for its sedative properties, which can be beneficial in managing migraine-related symptoms but may also lead to drowsiness as a side effect. The compound is typically administered in tablet form and is often prescribed for patients who experience frequent migraine attacks. Its mechanism of action involves the inhibition of vasodilation and the modulation of neurotransmitter release, which helps in alleviating migraine symptoms. As with any medication, it is essential to consider potential side effects, contraindications, and interactions with other drugs when prescribing or using pizotifen maleate.
Formula:C23H25NO4S
InChI:InChI=1/C19H21NS.C4H4O4/c1-20-11-8-15(9-12-20)19-16-5-3-2-4-14(16)6-7-18-17(19)10-13-21-18;5-3(6)1-2-4(7)8/h2-5,10,13H,6-9,11-12H2,1H3;1-2H,(H,5,6)(H,7,8)/b;2-1-
InChI key:InChIKey=GGYSHFFKUHGBIK-BTJKTKAUSA-N
SMILES:CN1CCC(=C2C3=C(CCC=4C2=CC=CC4)SC=C3)CC1.C(=C\C(O)=O)\C(O)=O
Synonyms:
  • Piperidine, 4-(9,10-dihydro-4H-benzo[4,5]cyclohepta[1,2-b]thien-4-ylidene)-1-methyl-, (2Z)-2-butenedioate (1:1)
  • Piperidine, 4-(9,10-dihydro-4H-benzo[4,5]cyclohepta[1,2-b]thien-4-ylidene)-1-methyl-, maleate (1:1)
  • Piperidine, 4-(9,10-dihydro-4H-benzo[4,5]cyclohepta[1,2-b]thien-4-ylidene)-1-methyl-, (Z)-2-butenedioate (1:1)
  • 4-(1-Methyl-4-piperidylidene)-9,10-dihydro-4H-benzo[4,5]cyclohepta[1,2-b]thiophene hydrogen maleate
  • 4-(9,10-Dihydro-4H-benzo(4,5)cyclohepta(1,2-b)thien-4-ylidene)-1-methylpiperidinium hydrogen maleate
  • Pizotifen maleate
  • 4H-Benzo[4,5]cyclohepta[1,2-b]thiophene, piperidine deriv.
  • 4-(9,10-dihydro-4H-benzo[4,5]cyclohepta[1,2-b]thiophen-4-ylidene)-1-methylpiperidinium (2Z)-3-carboxyprop-2-enoate
Sort by
The purity filter is not visible because current products do not have associated purity data for filtering.
Found 1 products.