CAS 252870-46-5

nAChR agonist 2

CAS: 252870-46-5

Compound 8, identified as a selective alpha4beta2 (α4β2) neuronal acetylcholine receptor (nAChR) agonist, demonstrates a dissociation constant (Kd) of 26 nM,

Formula: C₁₁H₁₆N₂

Color and Shape: Solid

Molecular weight: 176.263

Ref: TM-T40177

(E)-N-Methyl-4-(3-pyridinyl)-3-buten-1-amine oxalate

CAS: 252870-46-5

(E)-N-Methyl-4-(3-pyridinyl)-3-buten-1-amine oxalate is a research tool that is used to study the ion channels and their pharmacology. It inhibits the activity of potassium channels. The ligand binds to the receptor, which is an ion channel in the cell membrane. This binding activates or inhibits the receptor, leading to a change in membrane potential. The ligand may bind to any of these receptors: acetylcholine receptors, alpha adrenergic receptors, beta adrenergic receptors, GABA receptors, histamine H1 receptor, serotonin 5HT2A receptor, serotonin 5HT2C receptor, dopamine D2 receptor.

Formula: C₁₁H₁₆N₂

Purity: Min. 95%

Molecular weight: 176.26 g/mol

Ref: 3D-CKA87046