CAS 254964-60-8

Tasquinimod

Description:

Tasquinimod is a small molecule with the chemical formula C16H15N3O2, primarily recognized for its potential therapeutic applications, particularly in oncology. It functions as an immunomodulatory agent, influencing the immune system's response to cancer. Tasquinimod is known to inhibit tumor growth and metastasis by modulating the tumor microenvironment and enhancing anti-tumor immunity. Its mechanism of action involves the inhibition of angiogenesis and the alteration of immune cell activity, particularly affecting myeloid-derived suppressor cells. The compound is typically administered orally and has been investigated in clinical trials for various types of cancer, including prostate cancer. Tasquinimod's safety profile and pharmacokinetics have been subjects of research, contributing to its evaluation as a potential treatment option. As with many investigational drugs, ongoing studies aim to better understand its efficacy, optimal dosing, and long-term effects in cancer therapy.

Formula: C₂₀H₁₇F₃N₂O₄

InChI: InChI=1S/C20H17F3N2O4/c1-24(12-9-7-11(8-10-12)20(21,22)23)18(27)16-17(26)15-13(25(2)19(16)28)5-4-6-14(15)29-3/h4-10,26H,1-3H3

InChI key: InChIKey=ONDYALNGTUAJDX-UHFFFAOYSA-N

SMILES: OC=1C=2C(N(C)C(=O)C1C(N(C)C3=CC=C(C(F)(F)F)C=C3)=O)=CC=CC2OC

Synonyms:

• 1,2-Dihydro-4-hydroxy-5-methoxy-N,1-dimethyl-2-oxo-N-[4-(trifluoromethyl)phenyl]-3-quinolinecarboxamide
• 3-Quinolinecarboxamide, 1,2-dihydro-4-hydroxy-5-methoxy-N,1-dimethyl-2-oxo-N-[4-(trifluoromethyl)phenyl]-
• 4-Hydroxy-5-methoxy-N-methyl-1-methyl-2-oxo-N-(4-trifluoromethylphenyl)-1,2-dihydroquinoline-3-carboxamide
• Abr 215050
• Abr-5050
• N-Methyl-N-(4-trifluoromethylphenyl)-1,2-dihydro-4-hydroxy-5-methoxy-1-methyl-2-oxoquinoline-3-carboxamide
• Tasquinimod

Tasquinimod

CAS: 254964-60-8

Formula: C₂₀H₁₇F₃N₂O₄

Purity: 98%

Color and Shape: Solid

Molecular weight: 406.3552

Ref: IN-DA00BF4V

Tasquinimod

CAS: 254964-60-8

Tasquinimod

Purity: ≥98%

Molecular weight: 406.36g/mol

Ref: 54-BUP12222

Tasquinimod

CAS: 254964-60-8

Formula: C₂₀H₁₇F₃N₂O₄

Molecular weight: 406.36

Ref: 4Z-L-226006

Tasquinimod

CAS: 254964-60-8

Tasquinimod (ABR-215050) is an oral antiangiogenic agent and S100A9 inhibitor that binds to the HDAC4Zn2+ binding structural domain with Kd values ranging from 10 to 30 nM.Cost-effective and quality-assured.

Formula: C₂₀H₁₇F₃N₂O₄

Purity: 99.22% - >99.99%

Color and Shape: Solid

Molecular weight: 406.36

Ref: TM-T6695

TASQUINIMOD

CAS: 254964-60-8

Purity: 98%

Molecular weight: 406.3609924

Ref: 10-F799832

Tasquinimod

Controlled Product

CAS: 254964-60-8

Formula: C₂₀H₁₇F₃N₂O₄

Color and Shape: Neat

Molecular weight: 406.355

Ref: TR-T007820