CAS 2558-30-7

Desmethylflunitrazepam

Description:

Desmethylflunitrazepam, with the CAS number 2558-30-7, is a chemical compound that belongs to the benzodiazepine class of drugs. It is a derivative of flunitrazepam, which is known for its sedative and anxiolytic properties. Desmethylflunitrazepam is characterized by its ability to enhance the effects of the neurotransmitter gamma-aminobutyric acid (GABA) at the GABA-A receptor, leading to increased inhibitory neurotransmission in the central nervous system. This compound is typically encountered as a white to off-white crystalline powder and is soluble in organic solvents but has limited solubility in water. Its pharmacological effects include sedation, muscle relaxation, and anxiolysis, making it of interest in both medical and illicit contexts. However, due to its potential for abuse and dependence, desmethylflunitrazepam is subject to strict regulatory controls in many countries. Safety and toxicity profiles indicate that, like other benzodiazepines, it can lead to adverse effects, particularly when used in combination with other central nervous system depressants.

Formula:C₁₅H₁₀FN₃O₃

InChI:InChI=1/C15H10FN3O3/c16-12-4-2-1-3-10(12)15-11-7-9(19(21)22)5-6-13(11)18-14(20)8-17-15/h1-7H,8H2,(H,18,20)

InChI key:InChIKey=KNGIGRDYBQPXKQ-UHFFFAOYSA-N

SMILES:N(=O)(=O)C=1C=C2C(=NCC(=O)NC2=CC1)C3=C(F)C=CC=C3

Synonyms:

2H-1,4-Benzodiazepin-2-one, 5-(2-fluorophenyl)-1,3-dihydro-7-nitro-
2H-1,4-Benzodiazepin-2-one, 5-(o-fluorophenyl)-1,3-dihydro-7-nitro-
5-(2-fluorophenyl)-7-nitro-1,3-dihydro-2H-1,4-benzodiazepin-2-one
Demethylflunitrazepam
Desmethylflunitrazepam
Fonazepam
N-1-Desmethylflunitrazepam
N-Desmethylflunitrazepam
Norflunitrazepam
Ro 5-4435
5-(2-Fluorophenyl)-1,3-dihydro-7-nitro-2H-1,4-benzodiazepin-2-one
Desmethylflunitrazepam, Fonazepam
N-Desmethylflunitrazepam (CRM)
Flunitrazepan, N-desmethyl
N-DESMETHYLFLUNITRAZEPAM,100/MLINMETHANOL
N-DESMETHYLFLUNITRAZEPAM,1.0MG/MLINMETHANOL
N-Desmethylflunitrazepam solution
Ro-05-4435
N-DESMETHYLFLUNITRAZEPAM (100UG/ML METHANOL)
Nor-FlunitrazepaM 1.0 Mg/ML in Methanol
5-(2-Fluorphenyl)-1,3-dihydro-7-nitro-2H-1,4-benzodiazepin-2-on
Flunitrazepam EP Impurity B
See more synonyms

Purity (%)

100

Found 11 products.

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Desmethylflunitrazepam, 1mg/ml in Methanol
Controlled ProductPlease note that this is a controlled product in some countries, and needs to be treated in accordance with the relevant regulations. Be aware this might entail additional expenses and documentation.
CAS:
- 2558-30-7
Color and Shape:Single Solution
Ref: LP-FLU-71-1LM
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Desmethylflunitrazepam 1.0 mg/ml in Methanol
Controlled ProductPlease note that this is a controlled product in some countries, and needs to be treated in accordance with the relevant regulations. Be aware this might entail additional expenses and documentation.
CAS:
- 2558-30-7
Color and Shape:Single Solution
Ref: 61-AMP0069.02-01
1ml
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Desmethylflunitrazepam
Controlled ProductPlease note that this is a controlled product in some countries, and needs to be treated in accordance with the relevant regulations. Be aware this might entail additional expenses and documentation.
CAS:
- 2558-30-7
Color and Shape:Neat
Ref: 61-FOR0069.02
10mg
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Desmethylflunitrazepam 0.1 mg/ml in Methanol
Controlled ProductPlease note that this is a controlled product in some countries, and needs to be treated in accordance with the relevant regulations. Be aware this might entail additional expenses and documentation.
CAS:
- 2558-30-7
Color and Shape:Single Solution
Ref: 61-AMP0069.02-02
1ml
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Flunitrazepam EP Impurity B
Controlled ProductPlease note that this is a controlled product in some countries, and needs to be treated in accordance with the relevant regulations. Be aware this might entail additional expenses and documentation.
CAS:
- 2558-30-7
Formula:C₁₅H₁₀FN₃O₃
Color and Shape:Neat
Molecular weight:299.26
Ref: 86-MM0069.02
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Desmethylflunitrazepam
Controlled ProductPlease note that this is a controlled product in some countries, and needs to be treated in accordance with the relevant regulations. Be aware this might entail additional expenses and documentation.
CAS:
- 2558-30-7
Color and Shape:Neat
Ref: LP-FLU-71-10
10mg
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Nor-Flunitrazepam
Controlled ProductPlease note that this is a controlled product in some countries, and needs to be treated in accordance with the relevant regulations. Be aware this might entail additional expenses and documentation.
CAS:
- 2558-30-7
Applications A metabolite of Flunitrazepam (F500700). References Asai, H., et al.: J. Pharmacol. Exp. Ther., 277, 1004 (1996), Kilicarslan, T., et al.: Drug Metab. Dispos., 29, 460 (2001), Tanaka, E., et al.: J. Toxicol. Clin. Toxicol., 40, 69 (2002), 
Formula:C₁₅H₁₀FN₃O₃
Color and Shape:Yellow
Molecular weight:299.26
Ref: TR-N681050
10mg
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Nor-Flunitrazepam 1.0 mg/mL in Methanol
Controlled ProductPlease note that this is a controlled product in some countries, and needs to be treated in accordance with the relevant regulations. Be aware this might entail additional expenses and documentation.
CAS:
- 2558-30-7
Formula:C₁₅H₁₀FN₃O₃
Color and Shape:Single Solution
Molecular weight:299.26
Ref: TR-KIT0935
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5-(3-Fluorophenyl)-7-nitro-1,3-dihydro-1,4-benzodiazepin-2-one
Controlled ProductPlease note that this is a controlled product in some countries, and needs to be treated in accordance with the relevant regulations. Be aware this might entail additional expenses and documentation.
CAS:
- 2558-30-7
5-(3-Fluorophenyl)-7-nitro-1,3-dihydro-1,4-benzodiazepin-2-one is a potent inhibitor of the inflammatory response. It is a nonselective inhibitor of cyclooxygenase (COX) and lipoxygenase (LOX) that blocks the conversion of arachidonic acid to prostaglandins and leukotrienes. 5-(3-Fluorophenyl)-7-nitro-1,3-dihydro-1,4-benzodiazepin-2-one has been shown to inhibit COX activity in human serum and liver tissue samples. This compound also inhibits LOX activity in urine samples from patients with inflammatory diseases. It has been shown to exhibit single dose pharmacokinetic properties in healthy volunteers. The main metabolite of 5-(3-fluorophenyl)-7 nitro 1,3 di
Formula:C₁₅H₁₀FN₃O₃
Purity:Min. 95%
Color and Shape:Powder
Molecular weight:299.26 g/mol
Ref: 3D-FF96863
5mg
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10mg
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25mg
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Flunitrazepam EP Impurity B
CAS:
- 2558-30-7
Formula:C₁₅H₁₀FN₃O₃
Molecular weight:299.26
Ref: ST-EA-CP-F75002
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Desmethylflunitrazepam
CAS:
- 2558-30-7
Desmethylflunitrazepam (Norflunitrazepam) is a benzodiazepine derivative and an active metabolite of Flunitrazepam.
Formula:C₁₅H₁₀FN₃O₃
Color and Shape:Solid
Molecular weight:299.26
Ref: TM-T201723