CAS 26481-51-6: Tiprenolol

Description: Tiprenolol is a beta-adrenergic antagonist, primarily used in the treatment of glaucoma and ocular hypertension. As a non-selective beta-blocker, it works by reducing intraocular pressure through decreased aqueous humor production. The chemical structure of Tiprenolol includes a naphthalene ring, which contributes to its pharmacological properties. It is typically administered in the form of eye drops, allowing for localized action with minimal systemic absorption. The substance exhibits a moderate solubility in water, which is essential for its formulation as an ophthalmic solution. Tiprenolol's mechanism of action involves blocking beta-adrenergic receptors, leading to a reduction in heart rate and contractility, although its primary application is in eye care. Side effects may include ocular irritation, dry eyes, and systemic effects such as bradycardia or hypotension, particularly in sensitive individuals. Overall, Tiprenolol represents an important therapeutic option in managing conditions related to elevated intraocular pressure.

Formula: C₁₃H₂₁NO₂S

InChI: InChI=1S/C13H21NO2S/c1-10(2)14-8-11(15)9-16-12-6-4-5-7-13(12)17-3/h4-7,10-11,14-15H,8-9H2,1-3H3

InChI key: InChIKey=CSUNLSYSEQIDMO-UHFFFAOYSA-N

SMILES: OC(COC=1C=CC=CC1SC)CNC(C)C

Synonyms:

• 2-Propanol, 1-[(1-methylethyl)amino]-3-[2-(methylthio)phenoxy]-, (±)-
• 2-Propanol, 1-[(1-methylethyl)amino]-3-[2-(methylthio)phenoxy]-
• Tiprenolol
• 1-[(1-Methylethyl)amino]-3-[2-(methylthio)phenoxy]-2-propanol
• 2-Propanol, 1-(isopropylamino)-3-[o-(methylthio)phenoxy]-, (±)-

Tiprenolol

CAS: 26481-51-6

Tiprenolol is a beta adrenergic receptor antagonist.[1]

• Formula: C₁₃H₂₁NO₂S
• Purity: 99.43%
• Color and Shape: Solid
• Molecular weight: 255.38

1-[2-(Methylsulfanyl)phenoxy]-3-[(propan-2-yl)amino]propan-2-ol

CAS: 26481-51-6

Versatile small molecule scaffold

• Formula: C₁₃H₂₁NO₂S
• Purity: Min. 95%
• Molecular weight: 255.38 g/mol

1-[2-(methylsulfanyl)phenoxy]-3-[(propan-2-yl)amino]propan-2-ol

CAS: 26481-51-6

• Purity: 97%
• Molecular weight: 255.3800048828125