GPCR/G-Protein

Thrombin Receptor Activator for Peptide is also called Coagulation Factor II Receptor (1-5) or Proteinase …

UCSF924 is a potent and specific agonist of dopamine D4 receptor (DRD4) partial (EC50: 4.2 …

OPC 21268 is a non-peptide Arginine vasopressin(AVP) Receptor V antagonist.

SB408124 is a non-peptide antagonist for OX1 receptor with Ki of 57 nM and 27 …

Diacetolol D7 is deuterium-labeled diacetone Roller. Diacetol is the main metabolite of Acetolol. Diacetolol-adrenoceptor shielding …

Canagliflozin, a sodium-glucose transporter 2( SGLT2) and P-Glycoprotein inhibitor, is used in type 2 diabetes.

Islatravir is an effective anti-HIV-1 agent. It acting as a nucleoside reverse transcriptase inhibitor (EC50s: …

SB-334867 is a selective orexin-1 (OX1) receptor antagonist.

AZD4635 is a new-type adenosine 2A receptor (A2AR) inhibitor(Ki=1.7 nM).

Alpha-Methyldopa Sesquihydrate is a DOPA decarboxylase inhibitor and indirect 2-adrenergic receptor agonist used to treat …

Pimavanserin is an effective and specific serotonin 5-HT2A inverse agonist (pIC50: 8.73), used in the …

4'-O-Methylnyasol may have potential to be developed as medicines for the treatment of allergies by …

Felypressin is a synthetic analog of LYPRESSIN with a PHENYLALANINE substitution at residue 2. Felypressin …

1-Hydroxy-2,3,4,7-tetramethoxy-xanthone has vasodilatory action, it can cause vasodilation in the coronary artery pre-contracted with 1uM …

Semaglutide TFA is a agonist of glucagon-like peptide-1 (GLP-1) receptor,with a potential for type 2 …