GPCR/G-Protein
GPCR/G-Protein inhibitors are compounds that target G-protein coupled receptors (GPCRs) and associated G-proteins, which play critical roles in transmitting signals from the outside to the inside of cells. These inhibitors are essential for studying the signaling pathways mediated by GPCRs, which are involved in numerous physiological processes, including sensory perception, immune response, and neurotransmission. GPCR inhibitors are also important in drug development, as many therapeutic agents target these receptors. At CymitQuimica, we offer a wide range of high-quality GPCR/G-Protein inhibitors to support your research in pharmacology, cell biology, and related fields.
Subcategories of "GPCR/G-Protein"
- 5-HT Receptor(1,017 products)
- Adenosine Receptor(211 products)
- Adrenergic Receptor(3,154 products)
- Bombesin Receptor(34 products)
- Bradykinin Receptor(61 products)
- CXCR(159 products)
- CaSR(31 products)
- Cannabinoid Receptor(220 products)
- Cholecystokinin(1 products)
- Dopamine Receptor(445 products)
- Endothelin Receptor(85 products)
- GNRH Receptor(86 products)
- GPCR19(37 products)
- GRK(34 products)
- GTPase(23 products)
- Glucagon Receptor(197 products)
- Hedgehog/Smoothened(49 products)
- Histamine Receptor(389 products)
- LPA Receptor(21 products)
- Melatonin Receptor(26 products)
- OX Receptor(42 products)
- Opioid Receptor(330 products)
- PAFR(11 products)
- PKA(58 products)
- S1P Receptor(18 products)
- SGLT(30 products)
- Sigma receptor(48 products)
Show 19 more subcategories
Found 5839 products for "GPCR/G-Protein".
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Clonidine hydrochloride
CAS:Clonidine hydrochloride (Catapres) is a centrally active α-adrenergic agonist used predominantly as an antihypertensive agent.Formula:C9H10Cl3N3Purity:99.16% - 99.86%Color and Shape:SolidMolecular weight:266.55Cyproheptadine hydrochloride sesquihydrate
CAS:Cyproheptadine hydrochloride sesquihydrate (Peritol), an antihistamine, is an antagonist of serotonin and histamine2.Formula:C21H24ClNOPurity:99.77% - 99.99%Color and Shape:White SolidMolecular weight:341.88Lafutidine
CAS:Lafutidine (FRG-8813) is a newly developed histamine H(2)-receptor antagonist, which can inhibit gastric acid secretion.Formula:C22H29N3O4SPurity:99.96%Color and Shape:Yellowish White Crystalline PowderMolecular weight:431.55Upidosin
CAS:Upidosin (SB-216469), a uroselective α1 blocker: Ki α1a=0.34 nM, α1b=3.9 nM, α1d=1.5 nM, α2=33.3 nM.Formula:C31H33N3O4Purity:99.66%Color and Shape:SolidMolecular weight:511.61Rimonabant
CAS:Rimonabant (SR141716) is an inverse agonist for the cannabinoid receptor CB1.Formula:C22H21Cl3N4OPurity:98% - 99.91%Color and Shape:White SolidMolecular weight:463.79Metaproterenol hemisulfate
CAS:Metaproterenol hemisulfate (Orciprenaline sulfate) is a beta-2 adrenergic agonist used in the treatment of ASTHMA and BRONCHIAL SPASM.Formula:C11H17NO3·5H2O4SPurity:98.53% - 99.74%Color and Shape:White SolidMolecular weight:260.3AH 6809
CAS:AH 6809 blocks EP1, EP2, EP3, DP receptors (Ki: 1217-1597 nM human, 350 nM mouse EP2).Formula:C17H14O5Purity:97.59%Color and Shape:SolidMolecular weight:298.29Ref: TM-T14148
1mg34.00€5mg63.00€1mL*10mM (DMSO)67.00€10mg92.00€25mg165.00€50mg250.00€100mg401.00€200mg580.00€Nylidrin hydrochloride
CAS:Nylidrin HCl inhibits IgG1-induced histamine release in guinea pigs and IgE-induced release in rat mast cells & human basophils.Formula:C19H26ClNO2Purity:99.35%Color and Shape:White SolidMolecular weight:335.87Prucalopride
CAS:Prucalopride (R-93877), a selective 5-HT4A/4B agonist (Ki: 2.5/8 nM), is >290x more specific for these receptors.Formula:C18H26ClN3O3Purity:99.99% - >99.99%Color and Shape:White SolidMolecular weight:367.87Serazapine
CAS:Serazapine is a highly specific serotonin (5-HT2) binding inhibitor with anxiolytic activity for the treatment of anxiety disorders.Formula:C22H23N3O2Purity:99.29% - 99.97%Color and Shape:White SolidMolecular weight:361.44Fluparoxan hydrochloride
CAS:Fluparoxan hydrochloride is a highly selective and potent α2-adrenoceptor antagonist for the prevention, amelioration or treatment of neurodevelopmentalFormula:C10H11ClFNO2Purity:99.98%Color and Shape:SolidMolecular weight:231.65Aripiprazole
CAS:Aripiprazole (OPC-14597) is a piperazine/quinolone antipsychotic, partial agonist at 5-HT1A/D2, and antagonist at 5-HT2A.Formula:C23H27Cl2N3O2Purity:99.43% - 99.62%Color and Shape:White SolidMolecular weight:448.39Fluvoxamine maleate
CAS:Fluvoxamine maleate (DU-23000 (maleate)) is a selective serotonin reuptake inhibitor that is used in the treatment of depression and a variety of anxietyFormula:C19H25F3N2O6Purity:99.92% - 99.94%Color and Shape:White SolidMolecular weight:434.41Ref: TM-T1077
1mL*10mM (DMSO)35.00€10mg49.00€25mg65.00€50mg80.00€100mg109.00€200mg161.00€500mg263.00€Silodosin
CAS:Silodosin (KAD 3213) is an alpha-Adrenergic Blocker. The mechanism of action of silodosin is as an Adrenergic alpha-Antagonist.Formula:C25H32F3N3O4Purity:99.28% - 99.76%Color and Shape:White SolidMolecular weight:495.53Ref: TM-T1504
1500mgTo inquire5mg34.00€1mL*10mM (DMSO)35.00€10mg50.00€25mg73.00€50mg92.00€100mg99.00€200mg126.00€(3aR,9aR)-Fluparoxan
CAS:(3aR,9aR)-Fluparoxan is a highly selective and potent adrenergic receptor α2B antagonist for the prevention, amelioration or treatment of neurodevelopmentalFormula:C10H10FNO2Purity:97.82%Color and Shape:SolidMolecular weight:195.19Talastine
CAS:Talastine is an antihistamine compound that can induce an allergic rash.Formula:C19H21N3OPurity:99.44% - 99.84%Color and Shape:SolidMolecular weight:307.39Venlafaxine hydrochloride
CAS:Venlafaxine HCl, a cyclohexanol phenethylamine, acts as an SNRI antidepressant.Formula:C17H28ClNO2Purity:97.32% - 99.86%Color and Shape:SolidMolecular weight:313.86Roxatidine Acetate hydrochloride
CAS:Roxatidine Acetate hydrochloride (HOE 760) is a specific and competitive histamin H2-receptor antagonist. Roxatidine inhibits gastric acid secretion.Formula:C19H29ClN2O4Purity:99.49%Color and Shape:SolidMolecular weight:384.9Levosulpiride
CAS:Levosulpiride (S-(-)-Sulpiride) is the (S)-enantiomer of sulpiride, which is a D2 receptor antagonist, an atypical antipsychotic drug of the benzamide class.Formula:C15H23N3O4SPurity:98.20% - 99.88%Color and Shape:White SolidMolecular weight:341.439-Cyclopentyladenine
CAS:9-Cyclopentyladenine (NSC-19486) is an adenylate cyclase inhibitor that blocks cellular morphological differentiation and phosphorylation of specific signalingFormula:C10H13N5Purity:99.98%Color and Shape:White SolidMolecular weight:203.24
