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GPCR/G-Protein
K145 hydrochloride
CAS:
1449240-68-9
K145 is a specific inhibitor of SphK2 (IC50: 4.30 μM), while no inhibition of SphK1 …
Formula:
C18H25ClN2O3S
Purity:
98%
Molecular weight:
384.92
Ref: TM-TQ0138
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BETP
CAS:
1371569-69-5
BETP is an agonist of GLP-1 receptor (EC50s: 0.66 and 0.755 μM for human and …
Formula:
C20H17F3N2O2S
Purity:
98%
Molecular weight:
406.42
Ref: TM-TQ0124
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Lemborexant
CAS:
1369764-02-2
Lemborexant (E-2006) is a reversible and orally active dual antagonist of the orexin OX1 and …
Formula:
C22H20F2N4O2
Purity:
98%
Molecular weight:
410.42
Ref: TM-TQ0237
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Capadenoson
CAS:
544417-40-5
Capadenoson is a selective adenosine-A1 receptor agonist.
Formula:
C25H18ClN5O2S2
Purity:
98%
Molecular weight:
520.03
Ref: TM-TQ0125
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Tafluprost
CAS:
209860-87-7
Tafluprost, a prostaglandin analog, is the selective agonist of fluoroprostaglandin (FP) receptor PGF2α.
Formula:
C25H33F2O5
Purity:
98%
Molecular weight:
452.53
Ref: TM-TQ0203
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ONO-AE3-208
CAS:
402473-54-5
ONO-AE3-208 is an EP4 antagonist. It suppresses cell migration, invasion, and metastasis of prostate cancer.
Formula:
C24H21FN2O3
Purity:
98%
Molecular weight:
404.43
Ref: TM-TQ0290
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Avosentan
CAS:
290815-26-8
Avosentan (Ro 67-0565) is an effective and selective antagonist of the endothelin receptor (ETA receptor).
Formula:
C23H21N5O5S
Purity:
98%
Molecular weight:
479.51
Ref: TM-TQ0282
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GSK163090
CAS:
844903-58-8
GSK163090 is a specific and orally active 5-HT1A/B/D receptor antagonist (pKis: 9.4/8.5/9.7, and 6.3/6.7 for …
Formula:
C25H29N5O
Purity:
98%
Molecular weight:
415.53
Ref: TM-TQ0311
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GR 79236
CAS:
124555-18-6
GR79236 is an effective and selective adenosine A1 receptor agonist (Ki: 3.1 nM) that has …
Formula:
C15H17N5O5
Purity:
98%
Molecular weight:
351.36
Ref: TM-TQ0136
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PF-06291874
CAS:
1393124-08-7
PF-06291874 (Glucagon receptor antagonists-4) is a highly effective and orally active antagonist of the glucagon …
Formula:
C26H28F3N3O4
Purity:
98%
Molecular weight:
503.51
Ref: TM-TQ0239
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Bavisant
CAS:
929622-08-2
Bavisant (JNJ-31001074) is a selective and orally active antagonist of the human H3 receptor with …
Formula:
C19H27N3O2
Purity:
98%
Molecular weight:
329.44
Ref: TM-TQ0046
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Warangalone
CAS:
4449-55-2
Warangalone is an anti-malarial compound that can inhibit the growth of both strains of parasite …
Formula:
C25H24O5
Purity:
98%
Molecular weight:
404.46
Ref: TM-TQ0072
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MDA 19
CAS:
1048973-47-2
MDA 19 is a specific human CB2 receptor agonist (Ki: 43.3 nM).
Formula:
C21H23N3O2
Purity:
98%
Molecular weight:
349.43
Ref: TM-TQ0173
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BAR502
CAS:
1612191-86-2
BAR502 is a dual GPBAR1 and FXR agonist (IC50s: 0.4 μM and 2 μM).
Formula:
C25H40O3
Purity:
98%
Molecular weight:
392.62
Ref: TM-TQ0252
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Atrasentan hydrochloride
CAS:
195733-43-8
Atrasentan hydrochloride (ABT-627 hydrochloride) is an endothelin receptor antagonist (IC50: 0.0551 nM for ETA).
Formula:
C29H39ClN2O6
Purity:
98%
Molecular weight:
547.08
Ref: TM-TQ0270
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